The Journal of Organic Chemistry

Chemoselective Protection of Glutathione in the Preparation of Bioconjugates: The Case of Trypanothione Disulfide (Tue, 03 May 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00300
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Stereoselective Total Synthesis of (−)-Renieramycin T (Tue, 03 May 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00327
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Electrophilic Activation of P-Alkynes in the Synthesis of P-Substituted and P-Centered Heterocycles (Mon, 02 May 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00262
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Copper-Promoted Double Oxidative C–H Amination Cascade for the Synthesis of Imidazo[1,5-a]quinolines (Mon, 02 May 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00569
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Sulfinyl-Mediated Stereoselective Overman Rearrangements and Diels–Alder Cycloadditions (Fri, 29 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00365
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Low Band Gap Coplanar Conjugated Molecules Featuring Dynamic Intramolecular Lewis Acid–Base Coordination (Fri, 29 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00238
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A Photoinduced Cobalt-Catalyzed Synthesis of Pyrroles through in Situ-Generated Acylazirines (Fri, 29 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00511
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Palladium-Catalyzed Room-Temperature Acylative Suzuki Coupling of High-Order Aryl Borons with Carboxylic Acids (Fri, 29 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00421
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Stereoselective Formal Synthesis of (+)- and (−)-Cyclophellitol and (−)-Conduritol-B and Synthesis of (−)-Conduramine-B Derivative Using a Sulfinyl Moiety for C–O Bond Formation and α-Chloro Sulfide for C–C Bond Formation (Thu, 28 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00616
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Intramolecular Charge-Transfer Interaction of Donor–Acceptor–Donor Arrays Based on Anthracene Bisimide (Thu, 28 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00364
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Copper-Catalyzed Aza-Michael Addition of Aromatic Amines or Aromatic Aza-Heterocycles to α,β-Unsaturated Olefins (Thu, 28 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00341
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Dipolar Bent and Linear Acetylenes Substituted by Cationic Quinolinium and Anionic Benzoates. Formation of Mesomeric Betaines (Thu, 28 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00561
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Difunctionalization of Alkenes Using 1-Chloro-1,2-benziodoxol-3-(1H)-one (Thu, 28 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00295
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Stereocontrolled Construction of Tetrahydropyrano[2,3-c]pyrazole Scaffold via an Organocatalyzed Formal [3 + 3] Annulation (Thu, 28 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00196
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A Combined Experimental and Theoretical Approach to the Photogeneration of 5,6-Dihydropyrimidin-5-yl Radicals in Nonaqueous Media (Thu, 28 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00314
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Palladium-Catalyzed Deaminative Phenanthridinone Synthesis from Aniline via C–H Bond Activation (Thu, 28 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00378
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Synthesis of 9H-Pyrrolo[1,2-a]indole and 3H-Pyrrolizine Derivatives via a Phosphine-Catalyzed Umpolung Addition/Intramolecular Wittig Reaction (Thu, 28 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00473
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Ru(II)-Catalyzed Direct C(sp2)–H Activation/Selenylation of Arenes with Selenyl Chlorides (Thu, 28 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00634
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Ring-Opening of Donor–Acceptor Cyclopropanes by Boronic Acids and Potassium Organotrifluoroborates under Transition-Metal-Free Conditions (Thu, 28 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00320
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Enantioselective Synthesis of Ring-Fused Spiroannulated 1,2,3-Thiadiazole Derivatives (Thu, 28 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00127
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A One-Pot/Single-Analysis Approach to Substrate Scope Investigations Using Comprehensive Two-Dimensional Gas Chromatography (GC×GC) (Wed, 27 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00050
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A1/A2-Diamino-Substituted Pillar[5]arene-Based Acid–Base-Responsive Host–Guest System (Wed, 27 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00617
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Striking Difference between Succinimidomethyl and Phthalimidomethyl Radicals in Conjugate Addition to Alkylidenemalonate Initiated by Dimethylzinc (Tue, 26 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00485
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Chromene-Annulated Bacteriochlorins (Tue, 26 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00273
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Enantiomerically Pure [2.2]Paracyclophane-4-thiol: A Planar Chiral Sulfur-Based Building Block Readily Available by Resolution with an Amino Acid Chiral Auxiliary (Tue, 26 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00560
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A Hantzsch Amido Dihydropyridine as a Transfer Hydrogenation Reagent for α,β-Unsaturated Ketones (Tue, 26 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00041
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Regioselective Alkoxycarbonylation of Allyl Phenyl Ethers Catalyzed by Pd/dppb Under Syngas Conditions (Mon, 25 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00522
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The Synthesis of Methyl-Substituted Spirocyclic Piperidine-Azetidine (2,7-Diazaspiro[3.5]nonane) and Spirocyclic Piperidine-Pyrrolidine (2,8-Diazaspiro[4.5]decane) Ring Systems (Mon, 25 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b02890
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Lithium Enolates Derived from Pyroglutaminol: Aggregation, Solvation, and Atropisomerism (Mon, 25 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00459
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Chiral Bicyclic Bridgehead Phosphoramidite (Briphos) Ligands for Asymmetric Rhodium-Catalyzed 1,2- and 1,4-Addition (Mon, 25 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00033
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Preparation of 5-Aryl-2-Alkyltetrazoles with Aromatic Aldehydes, Alkylhydrazine, Di-tert-butyl Azodicarboxylate, and [Bis(trifluoroacetoxy)iodo]benzene (Mon, 25 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00606
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Total Synthesis of Brevisamide Using an Oxiranyl Anion Strategy (Fri, 22 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00484
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Enantioselective Organocatalytic Cyclopropanation of Enals Using Benzyl Chlorides (Fri, 22 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b02801
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The Reactivity of Thymine and Thymidine 5,6-Epoxides with Organometallic Reagents – A Route to Thymidine (6-4) Photoproduct Analogues (Fri, 22 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00495
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Regioselective Lithium–Iodine Exchange-Initiated Cleavage of 2-Iodomethyl-1,3-dioxanes: A Complex-Induced Proximity Effect (Fri, 22 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00496
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Palladium-Catalyzed Carbamate-Directed Regioselective Halogenation: A Route to Halogenated Anilines (Thu, 21 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00329
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Regioselectively Controlled Synthesis of N-Substituted (Trifluoromethyl)pyrimidin-2(1H)-ones (Thu, 21 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00382
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2,4,5-Trimethylimidazolium Scaffold for Anion Recognition Receptors Acting Through Charge-Assisted Aliphatic and Aromatic C–H Interactions (Thu, 21 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00468
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Engineering Light-Mediated Bistable Azobenzene Switches Bearing Urea d-Aminoglucose Units for Chiral Discrimination of Carboxylates (Wed, 20 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00200
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Construction of Stereogenic α,α-Disubstituted Cycloalkanones via 1° Amine Thiourea Dual Catalysis: Experimental Scope and Computational Analyses (Wed, 20 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00280
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Synthesis, Chemistry, and Photochemistry of Methylcyanobutadiyne in the Context of Space Science (Tue, 19 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00205
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Tetraphenylethene–2-Pyrone Conjugate: Aggregation-Induced Emission Study and Explosives Sensor (Tue, 19 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00267
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Total Synthesis of (−)-Luminacin D (Tue, 19 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00489
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Purely Chemical Approach for Preparation of d-α-Amino Acids via (S)-to-(R)-Interconversion of Unprotected Tailor-Made α-Amino Acids (Mon, 18 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b02707
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Chan–Evans–Lam Amination of Boronic Acid Pinacol (BPin) Esters: Overcoming the Aryl Amine Problem (Mon, 18 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00466
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Transition-Metal-Free Synthesis of N-Aryl Hydroxamic Acids via Insertion of Arynes (Fri, 15 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00111
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Synthesis of 1,2-Diketones via a Metal-Free, Visible-Light-Induced Aerobic Photooxidation of Alkynes (Fri, 15 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00097
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Correction to “Oxidation of Aryl Diphenylmethyl Sulfides Promoted by a Nonheme Iron(IV)-Oxo Complex: Evidence for an Electron Transfer-Oxygen Transfer Mechanism” (Fri, 15 Apr 2016)
The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00764
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Exploring the Application of the Negishi Reaction of HaloBODIPYs: Generality, Regioselectivity, and Synthetic Utility in the Development of BODIPY Laser Dyes (Thu, 14 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00350
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Complete Stereochemical Assignment of Campechic Acids A and B (Thu, 14 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00290
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Palladium-Catalyzed Ortho-Arylation of Carbamate-Protected Estrogens (Thu, 14 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00532
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Nickel-Catalyzed Phosphorylation of Phenol Derivatives via C–O/P–H Cross-Coupling (Thu, 14 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00289
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Three-Step Synthesis of Fluoranthenes through Pd-Catalyzed Inter- and Intramolecular C–H Arylation (Wed, 13 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00553
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Access to Isoquinolines and Isoquinolin-3-ols via Rh(III)-Catalyzed Coupling/Cyclization Cascade Reaction of Arylimidates and Diazo Compounds (Wed, 13 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00264
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N-Oxide as an Intramolecular Oxidant in the Baeyer–Villiger Oxidation: Synthesis of 2-Alkyl-2H-indazol-3-yl Benzoates and 2-Alkyl-1,2-dihydro-3H-indazol-3-ones (Wed, 13 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00251
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Why Do Enolate Anions Favor O-Alkylation over C-Alkylation in the Gas Phase? The Roles of Resonance and Inductive Effects in the Gas-Phase SN2 Reaction between the Acetaldehyde Enolate Anion and Methyl Fluoride (Tue, 12 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00351
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Synthesis of Functionalized 1,3,2-Benzodiazaborole Cores Using Bench-Stable Components (Tue, 12 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00435
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Conjugation, Substituent, and Solvent Effects on the Photogeneration of Quinone Methides (Tue, 12 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00331
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Silver(I)-Catalyzed Atroposelective Desymmetrization of N-Arylmaleimide via 1,3-Dipolar Cycloaddition of Azomethine Ylides: Access to Octahydropyrrolo[3,4-c]pyrrole Derivatives (Tue, 12 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00396
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Red to Near-Infrared Isoindole BODIPY Fluorophores: Synthesis, Crystal Structures, and Spectroscopic and Electrochemical Properties (Tue, 12 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00414
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One-Pot Synthesis of Benzo[4,5]imidazo[2,1-a]isoquinolines and Isoquinolino[3,4-b]quinoxalines via Tandem Cyclization Strategies (Tue, 12 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00338
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Hairpin Furans and Giant Biaryls (Tue, 12 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00492
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Controlled Reduction of Tertiary Amides to the Corresponding Alcohols, Aldehydes, or Amines Using Dialkylboranes and Aminoborohydride Reagents (Tue, 12 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00276
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Axially Chiral Bifunctional 8,8′-Biquinolyl: Synthesis of 7,7′-Dihydroxymethyl-8,8′-biquinolyl via Pd-Catalyzed Double C–H Oxidation of 7,7′-Dimethyl-8,8′-biquinolyl (Tue, 12 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00534
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Synthesis of 1,3-Disubstituted Imidazo[1,5-a]pyridines from Amino Acids via Catalytic Decarboxylative Intramolecular Cyclization (Mon, 11 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00343
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Comparative Reaction Diagrams for the SN2 Reaction Formulated According to the Leffler Analysis and the Hammond Postulate (Mon, 11 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00298
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Base-Mediated Cyclization Reaction of 2-(5-Hydroxy-1-pentynyl)benzonitriles to 4-Amino-2,3-dihydronaphtho[2,3-b]furanes and Synthesis of Furanonaphthoquinones (Mon, 11 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b02514
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Synthesis and Characterization of Two Unsymmetrical Indenofluorene Analogues: Benzo[5,6]-s-indaceno[1,2-b]thiophene and Benzo[5,6]-s-indaceno[2,1-b]thiophene (Fri, 08 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00340
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Silver(I)-Catalyzed Tandem Sigamatropic Rearrangement/1,3-H Shift/6π Aza-electrocyclization of N-Propargylic Hydrazones: A Mild Synthetic Route to 1,6-Dihydropyridazines (Fri, 08 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00428
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N2-Selective Iodofunctionalization of Olefins with NH-1,2,3-Triazoles to provide N2-Alkyl-Substituted 1,2,3-Triazoles (Fri, 08 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00185
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Enantioselective Recognition for Many Different Kinds of Chiral Guests by One Chiral Receptor Based on Tetraphenylethylene Cyclohexylbisurea (Fri, 08 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00371
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Gold(I)-Catalyzed Cascade Hydroarylation/Cycloaromatization to Indolizines via Pyridine Ring Construction (Fri, 08 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00346
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Diindenopyrenes: Extended 1,6- and 1,8-Pyrenoquinodimethanes with Singlet Diradical Characters (Fri, 08 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00389
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Discovery and Development of a Three-Component Oxidopyrylium [5 + 2] Cycloaddition (Fri, 08 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00394
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Tunable Push–Pull Interactions in 5-Nitrosopyrimidines (Thu, 07 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00446
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Stereoselective α-Hydroxylation of Amides Using Oppolzer’s Sultam as Chiral Auxiliary (Thu, 07 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00068
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Copper-Catalyzed C(sp2)–H Difluoroalkylation of Aldehyde Derived Hydrazones with Diboron as Reductant (Thu, 07 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00324
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Lewis Acid Catalyzed Friedel–Crafts Alkylation of Alkenes with Trifluoropyruvates (Thu, 07 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00358
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Enantioselective Synthesis of Dideoxy-tetrafluorinated Hexoses (Wed, 06 Apr 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b00302
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Regiospecifically Fluorinated Polycyclic Aromatic Hydrocarbons via Julia–Kocienski Olefination and Oxidative Photocyclization. Effect of Fluorine Atom Substitution on Molecular Shape (Tue, 22 Mar 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b02580
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Synthesis and Shuttling Behavior of [2]Rotaxanes with a Pyrrole Moiety (Sun, 20 Mar 2016)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b02911
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