The Journal of Organic Chemistry

Pd-Catalyzed Reigoselective Arylation on the C-5 Position of N-Aryl 1,2,3-Triazoles (Wed, 04 Mar 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/jo5026145
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Stereoselective Synthesis of the Diazonamide A Macrocyclic Core (Wed, 04 Mar 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/jo5029419
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The Aza-Wharton Reaction: Syntheses of Cyclic Allylic Amines and Vicinal Hydroxyamines from the Respective Acylaziridines (Wed, 04 Mar 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/jo5029387
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Effects of Thionation and Fluorination on Cis–Trans Isomerization in Tertiary Amides: An Investigation of N-Alkylglycine (Peptoid) Rotamers (Wed, 04 Mar 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00048
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Synthesis of Trifluoromethyl-Containing Vicinal Diamines by Asymmetric Decarboxylative Mannich Addition Reactions (Wed, 04 Mar 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00124
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Versatile Access to Martin’s Spirosilanes and Their Hypervalent Derivatives (Wed, 04 Mar 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/jo5028497
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Structure–Reactivity Relationship of Trifluoromethanesulfenates: Discovery of an Electrophilic Trifluoromethylthiolating Reagent (Tue, 03 Mar 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/jo502645m
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Enantioselective Assembly of Spirocyclic Oxindole-dihydropyranones through NHC-Catalyzed Cascade Reaction of Isatins with N-Hydroxybenzotriazole Esters of α,β-Unsaturated Carboxylic Acid (Tue, 03 Mar 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/jo502920w
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Anion Receptors Based on Halogen Bonding with Halo-1,2,3-triazoliums (Tue, 03 Mar 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00028
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Kinetic Resolution of α-Methylene-β-hydroxy Esters Catalyzed by Acyl Transfer Catalyst An-PIQ (Mon, 02 Mar 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00073
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Mechanistic Insight into the Dehydro-Diels–Alder Reaction of Styrene–Ynes (Mon, 02 Mar 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00200
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Stereoselective Synthesis of 3-Methyleneisoindolin-1-ones via Base-Catalyzed Intermolecular Reactions of Electron-Deficient Alkynes with N-Hydroxyphthalimides (Mon, 02 Mar 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00002
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Rhodium-Catalyzed 1,4-Addition of Arylboronic Acids to 3-Benzylidene-1H-pyrrolo[2,3-b]pyridin-2(3H)-one Derivatives (Mon, 02 Mar 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/jo502784h
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Rh(I)-Catalyzed Chemo- and Stereoselective Domino Cycloaddition of Optically Active Propargyl 2,4-Hexadienyl Ethers (Mon, 02 Mar 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00150
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Computational Mechanistic Study of the Julia–Kocieński Reaction (Fri, 27 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00008
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Silver-Catalyzed Double-Decarboxylative Cross-Coupling of α-Keto Acids with Cinnamic Acids in Water: A Strategy for the Preparation of Chalcones (Fri, 27 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/jo502642n
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Synthesis of 1,2-Borazaronaphthalenes from Imines by Base-Promoted Borylation of C–H bond (Fri, 27 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/jo5029437
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Brønsted Acid Catalyzed Asymmetric Diels–Alder Reactions: Stereoselective Construction of Spiro[tetrahydrocarbazole-3,3′-oxindole] Framework (Fri, 27 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00198
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Indium(III)-Catalyzed Knoevenagel Condensation of Aldehydes and Activated Methylenes Using Acetic Anhydride as a Promoter (Thu, 26 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00011
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Pd-Catalyzed Directed ortho-C–H Alkenylation of Phenylalanine Derivatives (Thu, 26 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/jo502912m
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Construction of Chiral α-Amino Quaternary Stereogenic Centers via Phase-Transfer Catalyzed Enantioselective α-Alkylation of α-Amidomalonates (Thu, 26 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/jo502791d
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Origin of High E-Selectivity in 4-Pyrrolidinopyridine-Catalyzed Tetrasubstituted α,α′-Alkenediol: A Computational and Experimental Study (Thu, 26 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/jo5029453
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Iridium-Catalyzed Direct Synthesis of Tryptamine Derivatives from Indoles: Exploiting N-Protected β-Amino Alcohols as Alkylating Agents (Thu, 26 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00195
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Synthesis of Substituted Resorcinol Monomethyl Ethers from 2-Bromo-3-methoxycyclohex-2-en-1-ones (Thu, 26 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00192
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Aminobenzofuran-Fused Rhodamine Dyes with Deep-Red to Near-Infrared Emission for Biological Applications (Thu, 26 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00077
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Taming Chlorine Azide: Access to 1,2-Azidochlorides from Alkenes (Thu, 26 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00009
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Synthesis of Quinolinones with Palladium-Catalyzed Oxidative Annulation between Acrylamides and Arynes (Wed, 25 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/jo5027673
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Base-Promoted Transannulation of Heterocyclic Enamines and 2,3-Epoxypropan-1-ones: Regio- and Stereoselective Synthesis of Fused Pyridines and Pyrroles (Wed, 25 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00067
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Light-Enabled Synthesis of Anhydrides and Amides (Wed, 25 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00003
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Photoremoval of Protecting Groups: Mechanistic Aspects of 1,3-Dithiane Conversion to a Carbonyl Group (Wed, 25 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/jo502953t
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χ-Shaped Bis(areno)-1,4-dihydropyrrolo[3,2-b]pyrroles Generated by Oxidative Aromatic Coupling (Wed, 25 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00052
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Cs2CO3-Promoted Carboxylation of N-Tosylhydrazones with Carbon Dioxide toward α-Arylacrylic Acids (Wed, 25 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/jo502908v
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Theoretical Examination of the S–C–P Anomeric Effect (Wed, 25 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/jo5029425
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Engaging Nonaromatic, Heterocyclic Tosylates in Reductive Cross-Coupling with Aryl and Heteroaryl Bromides (Wed, 25 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00135
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Reactivity and Stereoselectivity of 6π and Nazarov Electrocyclizations of Bridged Bicyclic Trienes and Divinyl Ketones (Tue, 24 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00070
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Dual Role of Acetanilides: Traceless Removal of a Directing Group through Deacetylation/Diazotation and Palladium-Catalyzed C–C-Coupling Reactions (Tue, 24 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00272
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Synthesis of Vinyl Trifluoromethyl Thioethers via Copper-Mediated Trifluoromethylthiolation of Vinyl Bromides (Tue, 24 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00144
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Preparation of Flavocoenzyme Isotopologues by Biotransformation of Purines (Tue, 24 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/jo502480w
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Synthesis of the β3-Adrenergic Receptor Agonist Solabegron and Analogous N-(2-Ethylamino)-β-amino Alcohols from O-Acylated Cyanohydrins – Expanding the Scope of Minor Enantiomer Recycling (Tue, 24 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00322
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Chemoenzymatic Routes to Enantiomerically Enriched and Polyoxygenated Perhydro-3,5a-methanoindeno[4,5-c]furans Related to the Tashironin Class of Sesquiterpenes (Tue, 24 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00303
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Reactivity-Based Dynamic Covalent Chemistry: Reversible Binding and Chirality Discrimination of Monoalcohols (Tue, 24 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/jo502801g
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Metal-Free Arylation of Ethyl Acetoacetate with Hypervalent Diaryliodonium Salts: An Immediate Access to Diverse 3-Aryl-4(1H)-Quinolones (Tue, 24 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/jo5023958
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Tools for Identifying Gelator Scaffolds and Solvents (Tue, 24 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/jo502915w
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Synthesis of Mimics of Pramanicin from Pyroglutamic Acid and Their Antibacterial Activity (Mon, 23 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/jo502810b
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Multicomponent Synthesis of Substituted and Fused-Ring Imidazoles via Phospha-münchnone Cycloaddition (Mon, 23 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/jo5028936
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Synthesis of 2-(3′-Indolyl)tetrahydrofurans by Oxidative Cycloetherification (Mon, 23 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00112
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Rhodium-Catalyzed Dehydrogenative Coupling of Phenylheteroarenes with Alkynes or Alkenes (Mon, 23 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00155
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Aza-Wacker-Type Reaction between Electron-Deficient Olefins and N-Alkylsulfonamides (Mon, 23 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/jo502823m
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Synthesis of 2-Aryl and 3-Aryl Benzo[b]furan Thioethers Using Aryl Sulfonyl Hydrazides as Sulfenylation Reagents (Fri, 20 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00146
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Synthesis, Functionalization, and Optical Properties of Chiral Carbazole-Based Diaza[6]helicenes (Fri, 20 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/jo5024188
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Electron-Deficient Heteroarenium Salts: An Organocatalytic Tool for Activation of Hydrogen Peroxide in Oxidations (Fri, 20 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/jo502865f
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Enantiomerically Pure 3-Aryl- and 3-Hetaryl-2-hydroxypropanoic Acids by Chemoenzymatic Reduction of 2-Oxo Acids (Fri, 20 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/jo502529g
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Platinum-Catalyzed Asymmetric Ring-Opening Reactions of Oxabenzonorbornadienes with Phenols (Fri, 20 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00065
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Diastereoselective Synthesis of Substituted Tetrahydrothiophenes and -thiopyrans via Thia-Prins Cyclization Reaction (Fri, 20 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/jo502831w
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Mechanistic Insights into a BINOL-Derived Phosphoric Acid-Catalyzed Asymmetric Pictet–Spengler Reaction (Thu, 19 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/jo5028134
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Copper-Catalyzed N-Cyanation of Sulfoximines by AIBN (Thu, 19 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/jo502607c
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Origins of Asymmetric Phosphazene Organocatalysis: Computations Reveal a Common Mechanism for Nitro- and Phospho-Aldol Additions (Thu, 19 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00063
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Synthesis of the Spirocyclic Framework of Sesterterpenoid Natural Products (Wed, 18 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/jo502897u
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A General Method for the One-Pot Reductive Functionalization of Secondary Amides (Wed, 18 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/jo502929x
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One-Pot Synthesis of Aryl Sulfones from Organometallic Reagents and Iodonium Salts (Tue, 17 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/jo5027518
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One-Pot Synthesis of Functionalized Benzo[b]thiophenes and Their Hetero-Fused Analogues via Intramolecular Copper-Catalyzed S-Arylation of In Situ Generated Enethiolates (Tue, 17 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00032
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Palladium-Catalyzed Aryl C(sp2)–H Bond Hydroxylation of 2-Arylpyridine Using TBHP as Oxidant (Tue, 17 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00167
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Preparation of Tetrasubstituted Olefins Using Mono or Double Aerobic Direct C–H Functionalization Strategies: Importance of Steric Effects (Mon, 16 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00148
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Ruthenium-Catalyzed Synthesis of 5-Amino-1,2,3-triazole-4-carboxylates for Triazole-Based Scaffolds: Beyond the Dimroth Rearrangement (Mon, 16 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/jo502577e
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Aerobic Palladium(II)-Catalyzed Dehydrogenative Heck Reaction in the Synthesis of Pyrenyl Fluorophores. A Photophysical Study of β-Pyrenyl Acrylates in Solution and in the Solid State (Mon, 16 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/jo502619k
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Cascade Arylalkylation of Activated Alkenes: Synthesis of Chloro- and Cyano-Containing Oxindoles (Mon, 16 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/jo502777b
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Synthesis of Unusual N-Acylated Aminosugar Fragments of Mycobacterium marinum Lipooligosaccharide IV (Mon, 16 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00064
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Catalyst-Free and Metal-Free Electrophilic Bromoamidation of Unactivated Olefins Using the N-Bromosuccinimide/Sulfonamide Protocol (Mon, 16 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/jo502416r
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Theoretical Study of Mechanism and Stereoselectivity of Catalytic Kinugasa Reaction (Fri, 13 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/jo502838p
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Synthesis of Enantiopure trans-2,5-Disubstituted Trifluoromethylpyrrolidines and (2S,5R)-5-Trifluoromethylproline (Fri, 13 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/jo502885v
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Selective Hydrogenation of Indolizines: An Expeditious Approach To Derive Tetrahydroindolizines and Indolizidines from Morita–Baylis–Hillman Adducts (Fri, 13 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/jo502471q
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One-Pot Synthesis of Multisubstituted Butyrolactonimidates: Total Synthesis of (−)-Nephrosteranic Acid (Fri, 13 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/jo5029166
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Palladium(II)-Catalyzed Sequential C–H Arylation/Aerobic Oxidative C–H Amination: One-Pot Synthesis of Benzimidazole-Fused Phenanthridines from 2-Arylbenzimidazoles and Aryl Halides (Fri, 13 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/jo502632b
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Possibility of [1,5] Sigmatropic Shifts in Bicyclo[4.2.0]octa-2,4-dienes (Thu, 12 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/jo5027639
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Stereoselective Formation of Eight-Membered Rings by Radical Cyclization of Silylenedioxy-Tethered Bis-methacrylate Derivatives (Thu, 12 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/jo502947k
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Transition-Metal-Free Access to Primary Anilines from Boronic Acids and a Common +NH2 Equivalent. (Thu, 12 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/jo5025078
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Total Synthesis of Cephalosporolide E via a Tandem Radical/Polar Crossover Reaction. The Use of the Radical Cations under Nonoxidative Conditions in Total Synthesis (Wed, 11 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/jo502757c
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Visible Light Mediated Cyclization of Tertiary Anilines with Maleimides Using Nickel(II) Oxide Surface-Modified Titanium Dioxide Catalyst (Wed, 11 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/jo502901h
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Potassium Thiocyanate as Source of Cyanide for the Oxidative α-Cyanation of Tertiary Amines (Wed, 11 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/jo502846c
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Pharmaceutical Process Chemistry: Evolution of a Contemporary Data-Rich Laboratory Environment (Mon, 09 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/jo502879m
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Chemo- and Stereoselective Synthesis of Fluorinated Enamides from Ynamides in HF/Pyridine: Second-Generation Approach to Potent Ureas Bioisosteres (Fri, 23 Jan 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/jo502699y
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Design and Synthesis of α-Carboxy Nucleoside Phosphonate Analogues and Evaluation as HIV-1 Reverse Transcriptase-Targeting Agents (Fri, 09 Jan 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/jo502549y
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