The Journal of Organic Chemistry

β-Selective C-Arylation of Diisobutylaluminum Hydride Modified 1,6-Anhydroglucose: Synthesis of Canagliflozin without Recourse to Conventional Protecting Groups (Fri, 24 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00601
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Deuteration of Aromatic Rings under Very Mild Conditions through Keto-Enamine Tautomeric Amplification (Thu, 23 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00539
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Chemoenzymatic Synthesis of 36S Isotopologues of Methionine and S-Adenosyl-l-methionine (Thu, 23 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00608
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Synthesis of SF5-Substituted Tetrapyrroles, Metalloporphyrins, BODIPYs, and Their Dipyrrane Precursors (Thu, 23 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00528
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Synthesis of Bench-Stable Diarylmethylium Tetrafluoroborates (Thu, 23 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00418
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Regioselective Metal-Free One-Pot Synthesis of Functionalized 2-Aminothiophene Derivatives (Thu, 23 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00488
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Palladium-Catalyzed Tandem Carbene Migratory Insertion and Intramolecular Cyclization: Synthesis of Chromeno[4,3-b]chromene Compounds (Thu, 23 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00500
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Regioselective Synthesis of 3-Bromoquinoline Derivatives and Diastereoselective Synthesis of Tetrahydroquinolines via Acid-Promoted Rearrangement of Arylmethyl Azides (Wed, 22 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00375
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Asymmetric Synthesis of Dihydronaphthoquinones Containing Adjacent Stereocenters via a Sulfa-Michael Addition Triggered Ring-Expansion Approach (Wed, 22 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00502
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Two Stepwise Synthetic Routes toward a Hetero[4]rotaxane (Wed, 22 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00627
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Regio- and Stereoselective Iodoacyloxylations of Alkynes (Wed, 22 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00250
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Fluorescent Dyes with Directly Connected Xanthone and Xanthene Units (Wed, 22 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00479
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Development and Application of α-Heteroatom Ketones in Asymmetric Michael Reaction with β-trans-Nitroalkenes (Wed, 22 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00013
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Chiral Recognition of Carboxylates by a Static Library of Thiourea Receptors with Amino Acid Arms (Wed, 22 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00403
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Iron/Copper Co-Catalyzed Synthesis of Vinyl Sulfones from Sulfonyl Hydrazides and Alkyne Derivatives (Wed, 22 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00558
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BF3-Mediated cis-Selective Cycloaddition of O-Silyloxime with Alkenes (Wed, 22 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00426
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Development of n-Type Semiconductor Based on Cyclopentene- or Cyclohexene-Fused [C60]-Fullerene Derivatives (Wed, 22 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00530
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Gold as Catalyst for the Hydroarylation and Domino Hydroarylation/N1–C4 Cleavage of β-Lactam-Tethered Allenyl Indoles (Tue, 21 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00535
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Ru(II)-Catalyzed β-Carboline Directed C–H Arylation and Isolation of Its Cycloruthenated Intermediates (Tue, 21 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00411
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Synthesis of Five-, Six-, and Seven-Membered 1,3- and 1,4-Heterocyclic Compounds via Intramolecular Hydroalkoxylation/Hydrothioalkoxylation of Alkenols/Thioalkenols (Mon, 20 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00049
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Regioselective Transition-Metal-Free Synthesis of 2-(Trimethylsilylmethylene)pyrrol-3-ones by Thermal Cyclization of Acetylenic Enamines (Mon, 20 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00398
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Mechanistic Investigation on the Formation of 2-Halo-3-aryl-4(3H)-quinazoliniminium Halides from Heteroenyne-allenes: A Computational Study (Mon, 20 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/jo502664s
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Synthesis toward CRHR1 Antagonists through 2,7-Dimethylpyrazolo[1,5-α][1,3,5]triazin-4(3H)-one C–H Arylation (Mon, 20 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/jo502894r
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Enantioselective Synthesis of (+)-Petromyroxol, Enabled by Rhodium-Catalyzed Denitrogenation and Rearrangement of a 1-Sulfonyl-1,2,3-Triazole (Mon, 20 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00399
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Copper-Catalyzed Radical Methylation/C–H Amination/Oxidation Cascade for the Synthesis of Quinazolinones (Mon, 20 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00191
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Design and Synthesis of Fluorinated Dendrimers for Sensitive 19F MRI (Mon, 20 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00294
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DMF Dimethyl Acetal as Carbon Source for α-Methylation of Ketones: A Hydrogenation–Hydrogenolysis Strategy of Enaminones (Mon, 20 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00084
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Enantioselective Total Syntheses of (+)-Hostmanin A, (−)-Linderol A, (+)-Methyllinderatin and Structural Reassignment of Adunctin E (Fri, 17 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00331
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3-Fluoroazetidinecarboxylic Acids and trans,trans-3,4-Difluoroproline as Peptide Scaffolds: Inhibition of Pancreatic Cancer Cell Growth by a Fluoroazetidine Iminosugar (Fri, 17 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00463
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Dynamic Behavior of N-Heterocyclic Carbene Boranes: Boron–Carbene Bonds in B,B-Disubstituted N,N-Dimethylimidazol-2-ylidene Boranes Have Substantial Rotation Barriers (Fri, 17 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00324
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Diastereoselective Synthesis of 1-Deoxygalactonojirimycin, 1-Deoxyaltronojirimycin, and N-Boc-(2S,3S)-3-Hydroxypipecolic Acid via Proline Catalyzed α-Aminoxylation of Aldehydes (Fri, 17 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00424
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Stereoselective Synthesis of Arylglycine Derivatives via Palladium-Catalyzed α-Arylation of a Chiral Nickel(II) Glycinate (Fri, 17 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00314
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Tribenzodecacyclene and Hexabenzodecacyclene (Fri, 17 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00551
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One-Pot, Three-Component Approach to the Synthesis of 3,4,5-Trisubstituted Pyrazoles (Fri, 17 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/jo502946g
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Synthesis of β-Amino-α,β-unsaturated Ketone Derivatives via Sequential Rhodium-Catalyzed Sulfur Ylide Formation/Rearrangement (Fri, 17 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00521
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Regioselective Synthesis of Highly Substituted Imidazoles via the Sequential Reaction of Allenyl Sulfonamides and Amines (Fri, 17 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00141
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One-Pot Synthesis of 2,5-Diaryl 1,3,4-Oxadiazoles via Di-tert-butyl Peroxide Promoted N-Acylation of Aryl Tetrazoles with Aldehydes (Fri, 17 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00207
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Near-Silence of Isothiocyanate Carbon in 13C NMR Spectra: A Case Study of Allyl Isothiocyanate (Fri, 17 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00080
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Pd(II)-Catalyzed Pyridine N-Oxides Directed Arylation of Unactivated Csp3–H Bonds (Fri, 17 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00489
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Cu-Catalyzed Consecutive Hydroxylation and Aerobic Oxidative Cycloetherification under Microwave Conditions: Entry to 2-Arylbenzofuran-3-carboxylic Acids (Thu, 16 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/jo502802k
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Chiral Gold Phosphate Catalyzed Tandem Hydroamination/Asymmetric Transfer Hydrogenation Enables Access to Chiral Tetrahydroquinolines (Thu, 16 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00153
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Biomimetic Synthesis of Two Salmahyrtisanes: Salmahyrtisol A and Hippospongide A (Thu, 16 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00420
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Modular Approach to Reductive Csp2–H and Csp3–H Silylation of Carboxylic Acid Derivatives through Single-Pot, Sequential Transition Metal Catalysis (Thu, 16 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00564
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Electronic Alteration on Oligothiophenes by o-Carborane: Electron Acceptor Character of o-Carborane in Oligothiophene Frameworks with Dicyano-Vinyl End-On Group (Thu, 16 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00336
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Glycosylation with 2-Acetamido-2-deoxyglycosyl Donors at a Low Temperature: Scope of the Non-Oxazoline Method (Wed, 15 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00138
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Synthesis of the Tetrasaccharide Repeating Unit from Acinetobacter baumannii Serogroup O18 Capitalizing on Phosphorus-Containing Leaving Groups (Wed, 15 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00139
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Selectfluor-Promoted Sequential Reactions via Allene Intermediates: Metal-Free Construction of Fused Polycyclic Skeletons (Wed, 15 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00261
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Radical Cyclization of Epoxy Vinyl- and Allylsulfones Promoted by Titanocene Chloride (Wed, 15 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00206
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Total Synthesis and Reassignment of the Structures of the Antimicrobial Lipodepsipeptides Circulocin γ and δ (Wed, 15 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00349
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o-Boronato- and o-Trifluoroborato–Phosphonium Salts Supported by l-α-Amino Acid Side Chain (Tue, 14 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00246
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Catalytic Chemical Amide Synthesis at Room Temperature: One More Step Toward Peptide Synthesis (Tue, 14 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00378
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The Stabilizing Role of the Intramolecular C–H···O Hydrogen Bond in Cyclic Amides Derived From α-Methylbenzylamine (Tue, 14 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00286
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Synthesis of a Tight Intramolecular OH···Olefin Interaction, Probed by IR, 1H NMR, and Quantum Chemistry (Tue, 14 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00470
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Enhanced Reactivity in Hydrogen Atom Transfer from Tertiary Sites of Cyclohexanes and Decalins via Strain Release: Equatorial C–H Activation vs Axial C–H Deactivation (Tue, 14 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00636
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Site-Specific Description of the Enhanced Recognition Between Electrogenerated Nitrobenzene Anions and Dihomooxacalix[4]arene Bidentate Ureas (Mon, 13 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00441
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Structure–Activity Relationships for Antibacterial to Antifungal Conversion of Kanamycin to Amphiphilic Analogues (Mon, 13 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00248
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Two-Photon Fluorescent Probes for Biological Mg2+ Detection Based on 7-Substituted Coumarin (Mon, 13 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/jo502775t
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Anilide Formation from Thioacids and Perfluoroaryl Azides (Mon, 13 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00240
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Total Syntheses of the Resorcylic Acid Lactone Neocosmosin A and Its Enantiomer (Mon, 13 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00590
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Chiral Surfactant-Type Catalyst: Enantioselective Reduction of Long-Chain Aliphatic Ketoesters in Water (Mon, 13 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00241
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Stereoselectivity in the Lewis Acid Mediated Reduction of Ketofuranoses (Mon, 13 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00419
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A Sequential Ugi Multicomponent/Cu-Catalyzed Azide–Alkyne Cycloaddition Approach for the Continuous Flow Generation of Cyclic Peptoids (Mon, 13 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00445
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Design and Synthesis of Labystegines, Hybrid Iminosugars from LAB and Calystegine, as Inhibitors of Intestinal α-Glucosidases: Binding Conformation and Interaction for ntSI (Mon, 13 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00342
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One-Pot Synthesis of 5-Amino-2,5-dihydro-1-benzoxepines: Access to Pharmacologically Active Heterocyclic Scaffolds (Mon, 13 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00583
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Extended Piperidine–Piperidinone Protein Interface Mimics (Mon, 13 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00300
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Understanding the Effects of Bidentate Directing Groups: A Unified Rationale for sp2 and sp3 C–H Bond Activations (Fri, 10 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00580
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Visible-Light-Mediated Radical Aryldifluoroacetylation of Alkynes with Ethyl Bromodifluoroacetate for the Synthesis of 3-Difluoroacetylated Coumarins (Fri, 10 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00305
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Phototautomerization in Pyrrolylphenylpyridine Terphenyl Systems (Fri, 10 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00275
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Total Synthesis of the Tetracyclic Indole Alkaloid Ht-13-B (Fri, 10 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00433
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Influence of Alkoxy Groups on Rates of Acetal Hydrolysis and Tosylate Solvolysis: Electrostatic Stabilization of Developing Oxocarbenium Ion Intermediates and Neighboring-Group Participation To Form Oxonium Ions (Thu, 09 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00338
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FeCl3-Mediated Synthesis of β-Alkynyl Ketones via Domino Nucleophilic-Substitution/Intramolecular-Cyclization/Reverse Claisen Condensation of N-Cyclohexyl Propargylamines and 1,3-Diketones (Thu, 09 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00281
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Modulation of Amide Bond Rotamers in 5-Acyl-6,7-dihydrothieno[3,2-c]pyridines (Thu, 09 Apr 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00205
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Origin of the Regioselective Reduction of Chlorins (Fri, 06 Mar 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00137
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Effects of Thionation and Fluorination on Cis–Trans Isomerization in Tertiary Amides: An Investigation of N-Alkylglycine (Peptoid) Rotamers (Wed, 04 Mar 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00048
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Mechanistic Insight into the Dehydro-Diels–Alder Reaction of Styrene–Ynes (Mon, 02 Mar 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00200
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Dual Role of Acetanilides: Traceless Removal of a Directing Group through Deacetylation/Diazotation and Palladium-Catalyzed C–C-Coupling Reactions (Tue, 24 Feb 2015)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.5b00272
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