ACS Medicinal Chemistry Letters



[ASAP] Extending Cross Metathesis To Identify Selective HDAC Inhibitors: Synthesis, Biological Activities, and Modeling (Fri, 17 May 2019)
TOC Graphic ACS Medicinal Chemistry Letters DOI: 10.1021/acsmedchemlett.8b00440
>> Read More

[ASAP] DMSO-Perturbing Assay for Identifying Promiscuous Enzyme Inhibitors (Thu, 16 May 2019)
TOC Graphic ACS Medicinal Chemistry Letters DOI: 10.1021/acsmedchemlett.9b00093
>> Read More

[ASAP] Identification of a RIP1 Kinase Inhibitor Clinical Candidate (GSK3145095) for the Treatment of Pancreatic Cancer (Thu, 16 May 2019)
TOC Graphic ACS Medicinal Chemistry Letters DOI: 10.1021/acsmedchemlett.9b00108
>> Read More

[ASAP] Thioimidate Bond Formation between Cardiac Troponin C and Nitrile-containing Compounds (Thu, 16 May 2019)
TOC Graphic ACS Medicinal Chemistry Letters DOI: 10.1021/acsmedchemlett.9b00168
>> Read More

[ASAP] Closing the Loop: Developing an Integrated Design, Make, and Test Platform for Discovery (Wed, 15 May 2019)
TOC Graphic ACS Medicinal Chemistry Letters DOI: 10.1021/acsmedchemlett.9b00095
>> Read More

[ASAP] Synthesis and Optimization of K<sub>v</sub>7 (KCNQ) Potassium Channel Agonists: The Role of Fluorines in Potency and Selectivity (Tue, 14 May 2019)
TOC Graphic ACS Medicinal Chemistry Letters DOI: 10.1021/acsmedchemlett.9b00097
>> Read More

[ASAP] Dendrigraft of Poly-<sc>l</sc>-lysine as a Promising Candidate To Reverse Heparin-based Anticoagulants in Clinical Settings (Mon, 13 May 2019)
TOC Graphic ACS Medicinal Chemistry Letters DOI: 10.1021/acsmedchemlett.9b00090
>> Read More

[ASAP] Development of a Platform To Enable Efficient Permeability Evaluation of Novel Organo-Peptide Macrocycles (Fri, 10 May 2019)
TOC Graphic ACS Medicinal Chemistry Letters DOI: 10.1021/acsmedchemlett.9b00036
>> Read More

[ASAP] Do Zebrafish Obey Lipinski Rules? (Fri, 10 May 2019)
TOC Graphic ACS Medicinal Chemistry Letters DOI: 10.1021/acsmedchemlett.9b00063
>> Read More

[ASAP] Identification of RIPK3 Type II Inhibitors Using High-Throughput Mechanistic Studies in Hit Triage (Wed, 08 May 2019)
TOC Graphic ACS Medicinal Chemistry Letters DOI: 10.1021/acsmedchemlett.9b00065
>> Read More

[ASAP] Discovery of a Lead Triphenylethanamine Cholesterol Ester Transfer Protein (CETP) Inhibitor (Mon, 06 May 2019)
TOC Graphic ACS Medicinal Chemistry Letters DOI: 10.1021/acsmedchemlett.9b00086
>> Read More

[ASAP] Unveiling the Importance of Amide Protons in CSP:ComD Interactions in <italic toggle="yes">Streptococcus pneumoniae</italic> (Fri, 03 May 2019)
TOC Graphic ACS Medicinal Chemistry Letters DOI: 10.1021/acsmedchemlett.9b00038
>> Read More

[ASAP] Correction to “Selective PPARd Modulators Improve Mitochondrial Function: Potential Treatment for Duchenne Muscular Dystrophy (DMD)” (Wed, 24 Apr 2019)
ACS Medicinal Chemistry Letters DOI: 10.1021/acsmedchemlett.9b00160
>> Read More