ACS Medicinal Chemistry Letters

Discovery of GSK2193874: An Orally Active, Potent, and Selective Blocker of Transient Receptor Potential Vanilloid 4 (Tue, 21 Mar 2017)
TOC Graphic ACS Medicinal Chemistry Letters DOI: 10.1021/acsmedchemlett.7b00094
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Development and Biological Evaluation of a Photoactivatable Small Molecule Microtubule-Targeting Agent (Tue, 21 Mar 2017)
TOC Graphic ACS Medicinal Chemistry Letters DOI: 10.1021/acsmedchemlett.6b00483
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Discovery of Antimalarial Azetidine-2-carbonitriles That Inhibit P. falciparum Dihydroorotate Dehydrogenase (Fri, 17 Mar 2017)
TOC Graphic ACS Medicinal Chemistry Letters DOI: 10.1021/acsmedchemlett.7b00030
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Opioid Receptor Activity and Analgesic Potency of DPDPE Peptide Analogues Containing a Xylene Bridge (Thu, 16 Mar 2017)
TOC Graphic ACS Medicinal Chemistry Letters DOI: 10.1021/acsmedchemlett.7b00044
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Antioxidant Properties of Novel Dimers Derived from Natural β-Elemene through Inhibiting H2O2-Induced Apoptosis (Wed, 15 Mar 2017)
TOC Graphic ACS Medicinal Chemistry Letters DOI: 10.1021/acsmedchemlett.7b00035
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Discovery of Highly Selective Inhibitors of the Immunoproteasome Low Molecular Mass Polypeptide 2 (LMP2) Subunit (Mon, 13 Mar 2017)
TOC Graphic ACS Medicinal Chemistry Letters DOI: 10.1021/acsmedchemlett.6b00496
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RITA Mimics: Synthesis and Mechanistic Evaluation of Asymmetric Linked Trithiazoles (Thu, 09 Mar 2017)
TOC Graphic ACS Medicinal Chemistry Letters DOI: 10.1021/acsmedchemlett.6b00488
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Discovery of [1,2,3]Triazolo[4,5-d]pyrimidine Derivatives as Novel LSD1 Inhibitors (Wed, 08 Mar 2017)
TOC Graphic ACS Medicinal Chemistry Letters DOI: 10.1021/acsmedchemlett.6b00423
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Discovery of Highly Potent 2-Sulfonyl-Pyrimidinyl Derivatives for Apoptosis Inhibition and Ischemia Treatment (Tue, 07 Mar 2017)
TOC Graphic ACS Medicinal Chemistry Letters DOI: 10.1021/acsmedchemlett.6b00489
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Small Molecule Lysyl Oxidase-like 2 (LOXL2) Inhibitors: The Identification of an Inhibitor Selective for LOXL2 over LOX (Mon, 06 Mar 2017)
TOC Graphic ACS Medicinal Chemistry Letters DOI: 10.1021/acsmedchemlett.7b00014
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INCB24360 (Epacadostat), a Highly Potent and Selective Indoleamine-2,3-dioxygenase 1 (IDO1) Inhibitor for Immuno-oncology (Mon, 06 Mar 2017)
TOC Graphic ACS Medicinal Chemistry Letters DOI: 10.1021/acsmedchemlett.6b00391
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X-ray Structure of the Carboplatin-Loaded Apo-Ferritin Nanocage (Thu, 02 Mar 2017)
TOC Graphic ACS Medicinal Chemistry Letters DOI: 10.1021/acsmedchemlett.7b00025
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The Ecstasy and Agony of Assay Interference Compounds (Tue, 28 Feb 2017)
ACS Medicinal Chemistry Letters DOI: 10.1021/acsmedchemlett.7b00056
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