ChemMedChem



Benzodioxane‐benzamides as antibacterial agents: Computational and SAR studies to evaluate the influence of the 7‐substitution in FtsZ interaction ()
ChemMedChem, Volume 0, Issue ja, -Not available-.
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Synthesis and Biological Evaluation of Five‐Atom‐Linker‐Based Arylpiperazine Derivatives with an Atypical Antipsychotic Profile ()
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Trifluoromethyl Dihydrothiazine‐Based β‐Secretase (BACE1) Inhibitors with Robust Central β‐Amyloid Reduction and Minimal Covalent Binding Burden ()
ChemMedChem, Volume 14, Issue 22, Page 1894-1910, November 20, 2019.
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Development of Amphipathic Antimicrobial Peptide Foldamers Based on Magainin 2 Sequence ()
ChemMedChem, Volume 14, Issue 22, Page 1911-1916, November 20, 2019.
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Design and Synthesis of Conformationally Constrained RORγt Inverse Agonists ()
ChemMedChem, Volume 14, Issue 22, Page 1917-1932, November 20, 2019.
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Oxidative Cyclization‐Induced Activation of a Phosphoinositide 3‐Kinase Inhibitor for Enhanced Selectivity of Cancer Chemotherapeutics ()
ChemMedChem, Volume 14, Issue 22, Page 1933-1939, November 20, 2019.
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Novel Hydrophilic Riminophenazines as Potent Antiprotozoal Agents ()
ChemMedChem, Volume 14, Issue 22, Page 1940-1949, November 20, 2019.
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Anticancer Activity of Electron‐Deficient Metal Complexes against Colorectal Cancer in vitro Models ()
ChemMedChem, Volume 14, Issue 22, Page 1887-1893, November 20, 2019.
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Front Cover: Mitochondria‐Targeting Selenophene‐Modified BODIPY‐Based Photosensitizers for the Treatment of Hypoxic Cancer Cells (ChemMedChem 22/2019) ()
ChemMedChem, Volume 14, Issue 22, Page 1878-1878, November 20, 2019.
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Mitochondria‐Targeting Selenophene‐Modified BODIPY‐Based Photosensitizers for the Treatment of Hypoxic Cancer Cells ()
ChemMedChem, Volume 14, Issue 22, Page 1879-1886, November 20, 2019.
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Quinoline‐Conjugated Ruthenacarboranes: Toward Hybrid Drugs with a Dual Mode of Action ()
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New Challenges in Drug Discovery – July 8–11, 2019, Vitoria‐Gasteiz, Spain ()
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Bivalent SMAC Mimetics for Treating Cancer by Antagonizing Inhibitor of Apoptosis Proteins ()
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Dual Farnesoid X Receptor/Soluble Epoxide Hydrolase Modulators Derived from Zafirlukast ()
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Synthesis of new Pyridoclax analogs: Insights into their druggability through investigation of their physicochemical properties and their interactions with membranes ()
ChemMedChem, Volume 0, Issue ja, -Not available-.
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Exploring the Molecular Mechanisms Underlying the in vitro Anticancer Effects of Multitarget‐Directed Hydrazone Ruthenium(II)–Arene Complexes ()
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Synthesis and Structure‐Activity Relationships of N‐(4‐Benzamidino)‐Oxazolidinones: Potent and Selective Inhibitors of Kallikrein‐Related Peptidase 6 ()
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2,2’‐Bipyridine‐Modified Tamoxifen: A Versatile Vector for Molybdacarboranes ()
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Discovery of Novel Biased Mu‐Opioid‐Receptor Agonists for the Treatment of Pain ()
ChemMedChem, Volume 0, Issue ja, -Not available-.
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The 12th AFMC International Medicinal Chemistry Symposium (AIMECS 2019) in Istanbul, Turkey ()
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Tracking Hidden Binding Pockets Along the Molecular Recognition Path of l‐Trp to Indoleamine 2,3‐Dioxygenase 1 ()
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Antibody Conjugation of a Chimeric BET Degrader Enables in vivo Activity ()
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Proline‐Rich Peptides with Improved Antimicrobial Activity against E. coli, K. Pneumoniae, and A. Baumannii ()
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Potential Therapeutic Effects of Mg/HCOOH Metal Organic Framework on Relieving Osteoarthritis ()
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Synthesis of Combretastatin‐A4 Carboxamidest that Mimic Sulfonyl Piperazines by a Molecular Hybridization Approach: in vitro Cytotoxicity Evaluation and Inhibition of Tubulin Polymerization ()
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Dual Escherichia coli DNA Gyrase A and B Inhibitors with Antibacterial Activity ()
ChemMedChem, Volume 0, Issue ja, -Not available-.
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Discovery and Pharmacophore Mapping of a Low‐Nanomolar Inhibitor of P. falciparum Growth ()
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Cell‐Based Optimization of Covalent Reversible Ketoamide Inhibitors Bridging the Unprimed to the Primed Site of the Proteasome β5 Subunit ()
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Exploring the Antiplasmodial 2‐Aminopyridines as Potential Antitrypanosomal Agents ()
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Structure−Activity Relationships of Cinnamate Ester Analogues as Potent Antiprotozoal Agents ()
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Poly[N‐(2‐hydroxypropyl)methacrylamide]‐Modified Magnetic γ‐F2O3 Nanoparticles Conjugated with Doxorubicin for Glioblastoma Treatment ()
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A Novel Class of N‐Sulfonyl and N‐Sulfamoyl Noscapine Derivatives that Promote Mitotic Arrest in Cancer Cells ()
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Flexible Fragment Growing Boosts Potency of Quorum Sensing Inhibitors against Pseudomonas aeruginosa Virulence ()
ChemMedChem, Volume 0, Issue ja, -Not available-.
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Synthesis and anticancer activity of tertiary amides of salinomycin and their C20‐oxo analogs ()
ChemMedChem, Volume 0, Issue ja, -Not available-.
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The Activity of Small Urea‐γ‐AApeptides Toward Gram‐Positive Bacteria ()
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Structure‐Based Design, Synthesis, and Biological Evaluation of Imidazo[4,5‐b]Pyridin‐2‐one‐Based p38 MAP Kinase Inhibitors: Part 2 ()
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Ligand‐ and Structure‐Based Approaches of Escherichia coli FabI Inhibition by Triclosan Derivatives: From Chemical Similarity to Protein Dynamics Influence ()
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Design and analysis of the 4‐anilino‐quin(az)oline kinase inhibition profiles of GAK/SLK/STK10 using quantitative structure activity relationships ()
ChemMedChem, Volume 0, Issue ja, -Not available-.
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