ChemMedChem



Rational Adaptation of L3MBTL1 Inhibitors to Create Small‐Molecule Cbx7 Antagonists ()
ChemMedChem, EarlyView.
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An angle on MK2 inhibition ‐ Optimization and evaluation of prevention of activation inhibitors ()
ChemMedChem, Volume 0, Issue ja, -Not available-.
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Conjugation Of Dasatinib With MHI‐148 Has A Significant Advan‐tageous Effect In Viability Assays For Glioblastoma Cells ()
ChemMedChem, Volume 0, Issue ja, -Not available-.
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Total Synthesis of the Endocannabinoid Uptake Inhibitor Guineensine and SAR Studies ()
ChemMedChem, Volume 0, Issue ja, -Not available-.
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2‐Phenyloxazole‐4‐carboxamide as new scaffold for selective inhibition of human monoamine oxidase B ()
ChemMedChem, Volume 0, Issue ja, -Not available-.
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Identification of Phenylpyrazolone Dimers as a New Class of Anti‐Trypanosoma cruzi Agents ()
ChemMedChem, Volume 0, Issue ja, -Not available-.
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Recent Developments in the Design of Mn‐ and Ru‐based Hybrid CO‐Releasing Molecules (HYCOs) ()
ChemMedChem, Volume 0, Issue ja, -Not available-.
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Experimental and Computational Evaluation of Piperonylic Acid Derived Hydrazones Bearing Isatin Moieties as Dual Inhibitors of Cholinesterases and Monoamine Oxidases ()
ChemMedChem, Volume 14, Issue 14, Page 1359-1376, July 17, 2019.
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Novel BQCA‐ and TBPB‐Derived M1 Receptor Hybrid Ligands: Orthosteric Carbachol Differentially Regulates Partial Agonism ()
ChemMedChem, Volume 14, Issue 14, Page 1349-1358, July 17, 2019.
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Computer‐Assisted Selective Optimization of Side‐Activities—from Cinalukast to a PPARα Modulator ()
ChemMedChem, Volume 14, Issue 14, Page 1343-1348, July 17, 2019.
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Substituted Aminoacetamides as Novel Leads for Malaria Treatment ()
ChemMedChem, Volume 14, Issue 14, Page 1329-1335, July 17, 2019.
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Fragment Growing to Design Optimized Inhibitors for Human Blood Group B Galactosyltransferase (GTB) ()
ChemMedChem, Volume 14, Issue 14, Page 1336-1342, July 17, 2019.
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Front Cover: Structural States of Hdm2 and HdmX: X‐ray Elucidation of Adaptations and Binding Interactions for Different Chemical Compound Classes (ChemMedChem 14/2019) ()
ChemMedChem, Volume 14, Issue 14, Page 1304-1304, July 17, 2019.
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The Design of Potent, Selective and Drug‐Like RGD αvβ1 Small‐Molecule Inhibitors Derived from non‐RGD α4β1 Antagonists ()
ChemMedChem, Volume 14, Issue 14, Page 1315-1320, July 17, 2019.
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Structural States of Hdm2 and HdmX: X‐ray Elucidation of Adaptations and Binding Interactions for Different Chemical Compound Classes ()
ChemMedChem, Volume 14, Issue 14, Page 1305-1314, July 17, 2019.
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Small‐Molecule Activators of Glucose‐6‐phosphate Dehydrogenase (G6PD) Bridging the Dimer Interface ()
ChemMedChem, Volume 14, Issue 14, Page 1321-1324, July 17, 2019.
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Combining 1,3‐Ditriazolylbenzene and Quinoline to Discover a New G‐Quadruplex‐Interactive Small Molecule Active against Cancer Stem‐Like Cells ()
ChemMedChem, Volume 14, Issue 14, Page 1325-1328, July 17, 2019.
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Allosteric Modulators of Potential Targets Related to Alzheimer’s Disease: a Review ()
ChemMedChem, Volume 0, Issue ja, -Not available-.
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Structure–Affinity Relationships of Fluorinated Spirocyclic σ2 Receptor Ligands with an Exocyclic Benzylamino Moiety ()
ChemMedChem, EarlyView.
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Structure and Energetics of Ligand–Fluorine Interactions with Galectin‐3 Backbone and Side‐Chain Amides: Insight into Solvation Effects and Multipolar Interactions ()
ChemMedChem, EarlyView.
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Azaaurones as potent antimycobacterial agents active against MDR‐ and XDR‐TB ()
ChemMedChem, Volume 0, Issue ja, -Not available-.
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Roles of the Conserved Amino Acid Residues in Reduced Human Defensin 5: Cysteine and Arginine Are Indispensable for Its Antibacterial Action and LPS Neutralization ()
ChemMedChem, EarlyView.
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­Optimization of LpxC Inhibitors for Antibacterial Activity and Cardiovascular Safety ()
ChemMedChem, Volume 0, Issue ja, -Not available-.
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Rational Design of Efficient Organic Phototherapeutic Agents via Perturbation Theory for Enhancing Anticancer Therapeutics ()
ChemMedChem, EarlyView.
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[18F]PRIMATX, a new positron emission tomography tracer for in vivo imaging of autotaxin in lung and tumour tissues ()
ChemMedChem, Volume 0, Issue ja, -Not available-.
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A Hydrogen Peroxide Activatable Gemcitabine Prodrug for the Selective Treatment of Pancreatic Ductal Adenocarcinoma ()
ChemMedChem, EarlyView.
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Synthesis of substituted 5’‐aminoadenosine derivatives and evaluation of their inhibitory potential towards CD73 ()
ChemMedChem, Volume 0, Issue ja, -Not available-.
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Probing 2H‐Indazoles as Template for SGK1, Tie2 and SRC Kinase Inhibitors ()
ChemMedChem, Volume 0, Issue ja, -Not available-.
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Synthesis of Nitrogen‐Containing Goniothalamin Analogues with Higher Cytotoxic Activity and Selectivity Against Cancer Cells ()
ChemMedChem, Volume 0, Issue ja, -Not available-.
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Combined Scaffold Evaluation and Systems‐Level Transcriptome‐Based Analysis for Accelerated Lead Optimization Reveals Ribosomal Targeting Spirooxindole Cyclopropanes ()
ChemMedChem, EarlyView.
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Synthesis and Study of Multifunctional Cyclodextrin–Deferasirox Hybrids ()
ChemMedChem, EarlyView.
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Stability and Efficiency of Mixed Aryl Phosphonate Prodrugs ()
ChemMedChem, Volume 0, Issue ja, -Not available-.
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