Organic letters



[ASAP] Direct Use of Carboxylic Acids in the Photocatalytic Hydroacylation of Styrenes To Generate Dialkyl Ketones (Thu, 21 Nov 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b03871
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[ASAP] Feet-to-Feet Connected Trisresorcinarenes (Thu, 21 Nov 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b03693
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[ASAP] Correction to A Case of Serendipity: Synthesis, Characterization, and Unique Chemistry of a Stable, Ring-Unsubstituted Aliphatic <italic toggle="yes">p</italic>-Quinone Methide (Wed, 20 Nov 2019)
Organic Letters DOI: 10.1021/acs.orglett.9b03951
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[ASAP] One-Pot Enantioselective Synthesis of 2-Pyrrolidinone Derivatives Bearing a Trifluoromethylated All-Carbon Quaternary Stereocenter (Wed, 20 Nov 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b03758
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[ASAP] High-Throughput Solid-Phase Building Block Synthesis for DNA-Encoded Libraries (Wed, 20 Nov 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b03553
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[ASAP] Oxalic Acid Monothioester for Palladium-Catalyzed Decarboxylative Thiocarbonylation and Hydrothiocarbonylation (Wed, 20 Nov 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b03701
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[ASAP] Morusalones A–D, Diels–Alder Adducts with 6/7/6/6/6/6 Hexacyclic Ring Systems as Potential PTP1B Inhibitors from Cell Cultures of <italic toggle="yes">Morus alba</italic> (Wed, 20 Nov 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b03664
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[ASAP] Magnesiate-Utilized/Benzyne-Mediated Approach to Indenopyridones from 2-Pyridones: An Attempt To Synthesize the Indenopyridine Core of Haouamine (Wed, 20 Nov 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b03806
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[ASAP] An Approach to Peri-Fused Heterocycles: A Metal-Mediated Cascade Carbonylative Cyclization/Dearomatic Diels–Alder Reaction (Wed, 20 Nov 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b03698
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[ASAP] Chiral Spiro Phosphoramide-Catalyzed Sulfa-Michael Addition/Enantioselective Protonation of Exocyclic Enones (Wed, 20 Nov 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b03615
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[ASAP] Asymmetric Total Synthesis Enables Discovery of Antibacterial Activity of Siladenoserinols A and H (Wed, 20 Nov 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b03857
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[ASAP] Accelerated Discovery in Photocatalysis by a Combined Screening Approach Involving MS Tags (Wed, 20 Nov 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b03936
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[ASAP] Network Analysis of Substituted Bullvalenes (Wed, 20 Nov 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b03737
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[ASAP] Synthesis of Heterocyclic Core-Expanded Bis-Naphthalene Tetracarboxylic Diimides (Wed, 20 Nov 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b03891
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[ASAP] Enantioselective Radical Ring-Opening Cyanation of Oxime Esters by Dual Photoredox and Copper Catalysis (Wed, 20 Nov 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b03970
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[ASAP] Divergent Reactivity in Cu<sup>II</sup>-Catalyzed Oxidative Coupling between Indole/Tryptamine Derivatives and ß-Arylacrylic Acids (Wed, 20 Nov 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b03697
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[ASAP] Gold(I)-Catalyzed Glycosylation with Glycosyl Ynenoates as Donors (Wed, 20 Nov 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b03851
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[ASAP] Photocatalytic <italic toggle="yes">E</italic> ? <italic toggle="yes">Z</italic> Isomerization of ß-Ionyl Derivatives (Wed, 20 Nov 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b03842
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[ASAP] Direct Catalytic Asymmetric Synthesis of Oxindole-Derived d-Hydroxy-ß-ketoesters by Aldol Reactions (Wed, 20 Nov 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b03527
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[ASAP] DNA-Compatible Diazo-Transfer Reaction in Aqueous Media Suitable for DNA-Encoded Chemical Library Synthesis (Wed, 20 Nov 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b03726
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[ASAP] Sequential Energy Transfer Catalysis: A Cascade Synthesis of Angularly-Fused Dihydrocoumarins (Wed, 20 Nov 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b03882
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[ASAP] Agelanemoechine, a Dimeric Bromopyrrole Alkaloid with a Pro-Angiogenic Effect from the South China Sea Sponge <italic toggle="yes">Agelas nemoechinata</italic> (Wed, 20 Nov 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b03683
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[ASAP] Electrochemical Synthesis of <italic toggle="yes">trans</italic>-2,3-Disubstituted Aziridines via Oxidative Dehydrogenative Intramolecular C(sp<sup>3</sup>)–H Amination (Wed, 20 Nov 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b03641
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[ASAP] Visible Light-Induced Amide Bond Formation (Tue, 19 Nov 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b03905
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[ASAP] Synthesis of <italic toggle="yes">cis</italic>-ß-Amidevinyl Benziodoxolones from the Ethynyl Benziodoxolone–Chloroform Complex and Sulfonamides (Tue, 19 Nov 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b03990
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[ASAP] Asymmetric Synthesis of Functionalized Phenylalanine Derivatives via Rh-Catalyzed Conjugate Addition and Enantioselective Protonation Cascade (Tue, 19 Nov 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b03666
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[ASAP] Ligand-Controlled Regiodivergent Silylation of Allylic Alcohols by Ni/Cu Catalysis for the Synthesis of Functionalized Allylsilanes (Tue, 19 Nov 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b03822
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[ASAP] An <italic toggle="yes">anti</italic>-Carbopalladation/Amination Cascade with Alkynes: Access to Tetrasubstituted Enamines and Pyrroles (Tue, 19 Nov 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b03625
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[ASAP] Mild Intramolecular Ring Opening of Oxetanes (Tue, 19 Nov 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b03810
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[ASAP] Multifunctional Catalytic Surface Design for Concerted Acceleration of One-Pot Hydrosilylation–CO<sub>2</sub> Cycloaddition (Tue, 19 Nov 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b03602
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[ASAP] Lewis-Acid-Mediated Thiocyano Semipinacol Rearrangement of Allylic Alcohols for Construction of a-Quaternary Center ß-Thiocyano Carbonyls (Tue, 19 Nov 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b03722
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[ASAP] Aqueous Base Promoted <italic toggle="yes">O</italic>-Difluoromethylation of Carboxylic Acids with TMSCF<sub>2</sub>Br: Bench-Top Access to Difluoromethyl Esters (Tue, 19 Nov 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b03604
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[ASAP] Carbene-Catalyzed Enantioselective Addition of Thioamides to Bromoenals for Access to Thiazinone Heterocycles (Tue, 19 Nov 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b03685
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[ASAP] Visible-Light-Induced Remote C(sp<sup>3</sup>)–H Pyridylation of Sulfonamides and Carboxamides (Mon, 18 Nov 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b03879
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[ASAP] Divergent Synthesis of Isoquinolone and Isocoumarin Derivatives by the Annulation of Benzoic Acid with <italic toggle="yes">N</italic>-Vinyl Amide (Mon, 18 Nov 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b03638
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[ASAP] Phosphoramidates as Steering Elements for Highly Selective Access to Complementary Imidazo[1,2-<italic toggle="yes">a</italic>]pyrimidine Isomers (Mon, 18 Nov 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b03702
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[ASAP] Oxidative Hydro-, Bromo-, and Chloroheptafluoroisopropylation of Unactivated Alkenes with Heptafluoroisopropyl Silver (Mon, 18 Nov 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b03705
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[ASAP] Site-Selective Modification of a-Amino Acids and Oligopeptides via Native Amine-Directed ?-C(sp<sup>3</sup>)-H Arylation (Mon, 18 Nov 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b03607
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[ASAP] A Direct, Chemo-, and Regioselective Cross-Coupling Reaction of Arenes via Sequential Directed <italic toggle="yes">ortho</italic> Cuprations and Oxidation (Mon, 18 Nov 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b03719
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[ASAP] Total Synthesis of (+)-<italic toggle="yes">epi</italic>-Condyfoline (Mon, 18 Nov 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b03762
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[ASAP] Enantioselective Aza-Reformatsky Reaction with Ketimines (Fri, 15 Nov 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b03669
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[ASAP] <italic toggle="yes">N</italic>-Methoxyamide: An Alternative Amidation Reagent in the Rhodium(III)-Catalyzed C–H Activation (Thu, 14 Nov 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b03357
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[ASAP] Total Synthesis and Stereochemical Reassignment of Citrafungin A (Thu, 14 Nov 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b03830
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[ASAP] Asymmetric Conjugate Addition of Ethylene Sulfonyl Fluorides to 3-Amido-2-oxindoles: Synthesis of Chiral Spirocyclic Oxindole Sultams (Thu, 14 Nov 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b03911
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[ASAP] Direct Hydrofluorination of Methallyl Alkenes Using a Methanesulfonic Acid/Triethylamine Trihydrofluoride Combination (Thu, 14 Nov 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b03950
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[ASAP] Construction of Multiple-Substituted Chiral Cyclohexanes through Hydrogenative Desymmetrization of 2,2,5-Trisubstituted 1,3-Cyclohexanediones (Thu, 14 Nov 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b03622
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[ASAP] Three-Component Aminoselenation of Arynes (Thu, 14 Nov 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b03789
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[ASAP] Nickel-Catalyzed Transformation of Diazoacetates to Alkyl Radicals Using Alcohol as a Hydrogen Source (Thu, 14 Nov 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b03610
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[ASAP] Enantioselective Gold-Catalyzed Pictet–Spengler Reaction (Thu, 14 Nov 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b03656
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[ASAP] LiHMDS-Promoted Palladium-Catalyzed Sonogashira Cross-Coupling of Aryl Fluorides with Terminal Alkynes (Thu, 14 Nov 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b03815
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