Organic letters



[ASAP] N-Heterocyclic Carbene Catalyzed Synthesis of Trisubstituted Epoxides via Tandem Amidation/Epoxidation Sequence (Thu, 09 Apr 2020)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.0c01017
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[ASAP] Copper-Catalyzed Functionalization of Aza-Aromatic Rings with Fluoroalcohols via Direct C(sp<sup>2</sup>)–H/C(sp<sup>3</sup>)–H Coupling Reactions (Wed, 08 Apr 2020)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.0c00797
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[ASAP] Pd-Catalyzed Oxidative Annulation of Aryl Ethers with Alkynes: Synthesis of Functionalized Spirocycles and Naphthalenes (Wed, 08 Apr 2020)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.0c00970
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[ASAP] Palladium-Catalyzed Direct Oxidative C–H Activation/Annulation for Regioselective Construction of <italic toggle="yes">N</italic>-Acylindoles (Wed, 08 Apr 2020)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.0c00877
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[ASAP] Direct Synthesis of Dibenzophospholes from Biaryls by Double C–P Bond Formation via Phosphenium Dication Equivalents (Tue, 07 Apr 2020)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.0c00944
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[ASAP] BF<sub>3</sub>-Catalyzed Skeletal Rearrangement of 7-En-2-ynones to <italic toggle="yes">endo</italic>-Type Cyclic Dienes (Tue, 07 Apr 2020)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.0c00949
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[ASAP] Time-Economical Radical Cascade Cyclization/Haloazidation of 1,6-Enynes: Construction of Highly Functional Succinimide Derivatives (Tue, 07 Apr 2020)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.0c00682
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[ASAP] Electroreductive 4-Pyridylation of Electron-deficient Alkenes with Assistance of Ni(acac)<sub>2</sub> (Tue, 07 Apr 2020)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.0c01014
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[ASAP] Overturning the Peribysin Family Natural Products Isolated from <italic toggle="yes">Periconia byssoides</italic> OUPS-N133: Synthesis and Stereochemical Revision of Peribysins A, B, C, F, and G (Tue, 07 Apr 2020)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.0c00857
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[ASAP] Computation-Guided Development of the “Click” <italic toggle="yes">ortho</italic>-Quinone Methide Cycloaddition with Improved Kinetics (Tue, 07 Apr 2020)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.0c00578
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[ASAP] Site-Selective C–H Functionalization–Sulfination Sequence to Access Aryl Sulfonamides (Tue, 07 Apr 2020)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.0c00982
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[ASAP] Regiodivergent Synthesis of Bis(4-oxycoumarin)-based Dioxabicycles: Exploration of [4 + 4] (Heterocyclo)reversion/addition and 1,5-Hydrogen Shift Photochromism (Tue, 07 Apr 2020)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.0c00904
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[ASAP] One-Pot Regiodirected Annulations for the Rapid Synthesis of p-Extended Oligomers (Tue, 07 Apr 2020)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.0c01043
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[ASAP] Diastereoselective Construction of Cyclopropane-Fused Tetrahydroquinolines via a Sequential [4 + 2]/[2 + 1] Annulation Reaction (Tue, 07 Apr 2020)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.0c00874
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[ASAP] Metal-Catalyzed Cyclotrimerization Reactions of Cyanamides: Synthesis of 2-Aryl-a-carbolines (Tue, 07 Apr 2020)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.0c00891
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[ASAP] Electrochemical Oxidative Dehydrogenative Phosphorylation of <italic toggle="yes">N</italic>-Heterocycles with P(O)–H Compounds in Imidazolium-Based Ionic Liquid (Tue, 07 Apr 2020)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.0c00814
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[ASAP] Catalytic Asymmetric Allylic Amination with Isatins, Sulfonamides, Imides, Amines, and <italic toggle="yes">N</italic>-Heterocycles (Tue, 07 Apr 2020)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.0c00936
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[ASAP] Identification of Brassicadiene, a Diterpene Hydrocarbon Attractive to the Invasive Stink Bug <italic toggle="yes">Bagrada hilaris</italic>, from Volatiles of Cauliflower Seedlings, <italic toggle="yes">Brassica oleracea</italic> var. <italic toggle="yes">botrytis</italic> (Mon, 06 Apr 2020)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.0c00707
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[ASAP] A Hg(OTf)<sub>2</sub>-Catalyzed Enolate Umpolung Reaction Enables the Synthesis of Coumaran-3-ones and Indolin-3-ones (Mon, 06 Apr 2020)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.0c01096
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[ASAP] Supramolecular Conformational Control of Aliphatic Oligoketones by Rotaxane Formation (Mon, 06 Apr 2020)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.0c01010
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[ASAP] Total Synthesis and Antitrypanosomal Activity of Janadolide and Simplified Analogues (Mon, 06 Apr 2020)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.0c00840
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[ASAP] When Gold Meets Perfumes: Synthesis of Olfactive Compounds via Gold-Catalyzed Cycloisomerization Reactions (Mon, 06 Apr 2020)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.0c00843
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[ASAP] Total Synthesis of (±)-Thebainone A by Intramolecular Nitrone Cycloaddition (Mon, 06 Apr 2020)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.0c00905
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[ASAP] Multistep Photoisomerization of Dimesitylboron-Functionalized Stilbene Analogues (Mon, 06 Apr 2020)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.0c01042
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[ASAP] Three-Component Borylallenylation of Alkynes: Access to Densely Boryl-Substituted Ene-allenes (Mon, 06 Apr 2020)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.0c00643
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[ASAP] Zinc-Catalyzed Phosphonylation of Alcohols with Alkyl Phosphites (Mon, 06 Apr 2020)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.0c00932
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[ASAP] Rapid Access to Borylated Thiophenes Enabled by Visible Light (Fri, 03 Apr 2020)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.0c01076
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[ASAP] Highly Stereoselective Synthesis of 1,2-Disubstituted Indanes by Pd-Catalyzed Heck/Suzuki Sequence of Diarylmethyl Carbonates (Fri, 03 Apr 2020)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.0c00945
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[ASAP] Gold-Catalyzed Oxidative Cascade Cyclization of 1,3-Diynamides: Polycyclic N-Heterocycle Synthesis via Construction of a Furopyridinyl Core (Fri, 03 Apr 2020)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.0c01086
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[ASAP] Synthesis of Bridged Azacycles and Propellanes via Nitrene/Alkyne Cascades (Fri, 03 Apr 2020)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.0c00798
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[ASAP] Photoredox-Assisted Gold-Catalyzed Arylative Alkoxycyclization of 1,6-Enynes (Fri, 03 Apr 2020)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.0c00799
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[ASAP] Enzyme-Catalyzed Azepinoindole Formation in Clavine Alkaloid Biosynthesis (Fri, 03 Apr 2020)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.0c01132
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[ASAP] Construction of Thiazole-Fused Dihydropyrans via Formal [4 + 2] Cycloaddition Reaction on DNA (Fri, 03 Apr 2020)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.0c01016
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[ASAP] Nickel-Catalyzed Formal Aminocarbonylation of Unactivated Alkyl Iodides with Isocyanides (Fri, 03 Apr 2020)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.0c01022
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[ASAP] Toward FAIRness and a User-Friendly Repository for Supporting NMR Data (Fri, 03 Apr 2020)
Organic Letters DOI: 10.1021/acs.orglett.0c01143
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[ASAP] Clickable Bambusurils to Access Multivalent Architectures (Fri, 03 Apr 2020)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.0c00856
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[ASAP] Iridium-Catalyzed Direct C–H Amidation Producing Multicolor Fluorescent Molecules Emitting Blue-to-Red Light and White Light (Fri, 03 Apr 2020)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.0c00618
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[ASAP] Superelectrophilic Fe(III)–Ion Pairs as Stronger Lewis Acid Catalysts for (<italic toggle="yes">E</italic>)-Selective Intermolecular Carbonyl–Olefin Metathesis (Fri, 03 Apr 2020)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.0c00917
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[ASAP] Cascade Claisen and Meinwald Rearrangement for One-Pot Divergent Synthesis of Benzofurans and 2<italic toggle="yes">H</italic>-Chromenes (Fri, 03 Apr 2020)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.0c00770
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[ASAP] Ni-Catalyzed Allylic Dearomatization Reaction of ß-Naphthols with Allylic Alcohols (Fri, 03 Apr 2020)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.0c01109
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[ASAP] Synthesis of Hexahydropyridazines by [4 + 2] Cycloaddition of Donor–Acceptor Cyclobutanes and <italic toggle="yes">cis</italic>-Diazenes (Fri, 03 Apr 2020)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.0c00896
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[ASAP] Rhodium(III)-Catalyzed Asymmetric C–H Activation of <italic toggle="yes">N</italic>-Methoxybenzamide with Quinone and Its Application in the Asymmetric Synthesis of a Dihydrolycoricidine Analogue (Thu, 02 Apr 2020)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.0c01002
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[ASAP] Unexpected <italic toggle="yes">ortho</italic>-Heck Reaction under the Catellani Conditions (Thu, 02 Apr 2020)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.0c00952
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[ASAP] Selenacalix[4]selenophene: Synthesis, Structure, and Gel Formation of Cyclic Selenoether of Selenophene (Thu, 02 Apr 2020)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.0c00839
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[ASAP] Photocatalytic [2 + 2] Cycloaddition in DNA-Encoded Chemistry (Thu, 02 Apr 2020)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.0c00574
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[ASAP] Construction of Silicon-Containing Seven-Membered Rings by Catalytic [4 + 2 + 1] Cycloaddition through Rhodium Silylenoid (Thu, 02 Apr 2020)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.0c00690
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[ASAP] Alternarin A, a Drimane Meroterpenoid, Suppresses Neuronal Excitability from the Coral-Associated Fungi <italic toggle="yes">Alternaria</italic> sp. ZH-15 (Thu, 02 Apr 2020)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.0c00746
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[ASAP] Palladium-Catalyzed Mizoroki–Heck Reaction of Nitroarenes and Styrene Derivatives (Thu, 02 Apr 2020)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.0c00983
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[ASAP] K<sub>2</sub>CO<sub>3</sub>-Catalyzed Synthesis of 2,5-Dialkyl-4,6,7-tricyano-Decorated Indoles via Carbon–Carbon Bond Cleavage (Thu, 02 Apr 2020)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.0c01057
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[ASAP] Diisobutylaluminum Hydride Promoted Selectivity-Switchable Synthesis of Benzothiophene Oxides and Benzothiophenes via an Al–Li-Dimetalated Intermediate (Thu, 02 Apr 2020)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.0c00884
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