Organic letters



[ASAP] Rhodium(III)-Catalyzed Intramolecular Olefin Hydroarylation of Aromatic Aldehydes Using a Transient Directing Group (Fri, 17 May 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b01101
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[ASAP] Highly Regio- and Enantioselective Dienylation of <italic toggle="yes">p</italic>-Quinone Methides Enabled by an Organocatalyzed Isomerization/Addition Cascade of Allenoates (Fri, 17 May 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b01110
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[ASAP] Visible-Light Induced Radical Perfluoroalkylation/Cyclization Strategy To Access 2-Perfluoroalkylbenzothiazoles/Benzoselenazoles by EDA Complex (Fri, 17 May 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b01175
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[ASAP] Targeted Gene Inactivations Expose Silent Cytochalasans in <italic toggle="yes">Magnaporthe grisea</italic> NI980 (Fri, 17 May 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b01344
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[ASAP] Toward Acetylene Renaissance: Functionally Rich <italic toggle="yes">N</italic>-Aminoindoles from Acetylene Gas, Ketones, and Hydrazines in Two Steps (Fri, 17 May 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b01452
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[ASAP] Regio- and Enantioselective Synthesis of 1,2-Diamine Derivatives by Copper-Catalyzed Hydroamination (Fri, 17 May 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b01592
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[ASAP] Remote 1,5-Stereoselectivity Control by an <italic toggle="yes">N</italic>-Ligand Switch in the Pd(0)/InI-Promoted Reactions of 4-Ethynyl-ß-lactams with Aldehydes (Thu, 16 May 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b00891
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[ASAP] Ruthenium(VIII)-Catalyzed <italic toggle="yes">ipso</italic>-Dearomative Spiro-Etherification and Spiro-Amidation of Phenols (Thu, 16 May 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b01322
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[ASAP] Visible-Light-Triggered Cyanoalkylation of <italic toggle="yes">para</italic>-Quinone Methides and Its Application to the Synthesis of GPR40 Agonists (Thu, 16 May 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b01325
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[ASAP] H<sub>2</sub>O-Regulated Chemoselectivity in Oxa- Versus Aza-Michael Reactions (Thu, 16 May 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b01342
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[ASAP] [3 + 2]-Cycloaddition of 2<italic toggle="yes">H</italic>-Azirines with Nitrosoarenes: Visible-Light-Promoted Synthesis of 2,5-Dihydro-1,2,4-oxadiazoles (Thu, 16 May 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b01416
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[ASAP] Synthesis of a-Fluorinated Imides via Direct Fluorohydroxylation of Ynamides (Thu, 16 May 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b01428
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[ASAP] 2-Position-Selective Trifluoromethylthiolation of Six-Membered Heteroaromatic Compounds (Thu, 16 May 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b01474
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[ASAP] Switchable Skeletal Rearrangement of Dihydroisobenzofuran Acetals with Indoles (Thu, 16 May 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b01488
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[ASAP] Correction to Fischer Carbene Catalysis of Alkynol Cycloisomerization: Application to the Synthesis of the Altromycin B Disaccharide (Wed, 15 May 2019)
Organic Letters DOI: 10.1021/acs.orglett.9b01023
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[ASAP] Involvement of Peptide Epimerization in Poly-?-glutamic Acid Biosynthesis (Wed, 15 May 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b01121
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[ASAP] Catalytic Cascade Reaction To Access Cyclopentane-Fused Heterocycles: Expansion of Pd–TMM Cycloaddition (Wed, 15 May 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b01178
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[ASAP] Catalytic Diastereo- and Enantioselective Synthesis of 2-Imidazolinones (Wed, 15 May 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b01244
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[ASAP] Gold(I)-Catalyzed Oxidation of Acyl Acetylenes to Vicinal Tricarbonyls (Wed, 15 May 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b01297
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[ASAP] Metal-Free Denitrogenative C–C Couplings of Pyridotriazoles with Boronic Acids To Afford a-Secondary and a-Tertiary Pyridines (Wed, 15 May 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b01334
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[ASAP] Tunable <italic toggle="yes">E</italic>–<italic toggle="yes">Z</italic> Photoisomerization in a,ß-Peptide Foldamers Featuring Multiple (<italic toggle="yes">E</italic>/<italic toggle="yes">Z</italic>)-3-Aminoprop-2-enoic Acid Units (Wed, 15 May 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b01360
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[ASAP] Ligand-Accelerated Iron Photocatalysis Enabling Decarboxylative Alkylation of Heteroarenes (Wed, 15 May 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b01439
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[ASAP] Regioselective Intermolecular Sulfur–Oxygen Difunctionalization (Phenoxysulfonylation) of Alkynes: One-Pot Construction of (<italic toggle="yes">Z</italic>)-ß-Phenoxy Vinylsulfones (Tue, 14 May 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b01041
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[ASAP] Desulfurization of Diaryl(heteroaryl) Sulfoxides with Benzyne (Tue, 14 May 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b01144
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[ASAP] Diazocine Derivatives: A Family of Azobenzenes for Photochromism with Highly Enhanced Turn-On Fluorescence (Tue, 14 May 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b01215
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[ASAP] Synthesis of Substituted Benzaldehydes via a Two-Step, One-Pot Reduction/Cross-Coupling Procedure (Tue, 14 May 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b01274
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[ASAP] A Synthesis of Multifunctionalized Indoles from [3 + 2] Annulation of 2-Bromocyclopropenes with Anilines (Tue, 14 May 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b01276
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[ASAP] Euphorkanlide A, a Highly Modified Ingenane Diterpenoid with a C<sub>24</sub> Appendage from <italic toggle="yes">Euphorbia kansuensis</italic> (Tue, 14 May 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b01315
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[ASAP] Correction to Synthesis of Enantioenriched a-Chiral Bicyclo[1.1.1]pentanes (Tue, 14 May 2019)
Organic Letters DOI: 10.1021/acs.orglett.9b01503
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[ASAP] Sodium-Catalyzed Friedel–Crafts Reactions and Mechanistic Insight (Mon, 13 May 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b00747
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[ASAP] Access to 3-Deazaguanosine Building Blocks for RNA Solid-Phase Synthesis Involving Hartwig–Buchwald C–N Cross-Coupling (Mon, 13 May 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b00855
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[ASAP] Synthesis of Hydroxyisooxophlorins by Oxidative Degradation of <italic toggle="yes">meso</italic>-Hydroxyporphyrins (Mon, 13 May 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b01066
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[ASAP] Potassium Alkylpentafluorosilicates, Primary Alkyl Radical Precursors in the C-1 Alkylation of Tetrahydroisoquinolines (Mon, 13 May 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b01124
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[ASAP] Synthesis of ß-Amino Diaryldienones Using the Mannich Reaction (Mon, 13 May 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b01195
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[ASAP] Trapping of Zwitterionic Intermediates by Isatins and Imines: Synthesis of Benzoxazines Bearing a C4-Quaternary Stereocenter (Mon, 13 May 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b01207
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[ASAP] Cobalt Catalyzed Hydroarylation of Michael Acceptors with Indolines Directed by a Weakly Coordinating Functional Group (Mon, 13 May 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b01228
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[ASAP] Porous Organic Polymer-Derived Nanopalladium Catalysts for Chemoselective Synthesis of Antitumor Benzofuro[2,3-<italic toggle="yes">b</italic>]pyrazine from 2-Bromophenol and Isonitriles (Mon, 13 May 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b01230
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[ASAP] Photocatalytic 1,1-Hydrofluoroalkylation of Alkynes with a Concurrent Vicinal Acylation: An Access to Fluoroalkylated Cyclic Ketones (Mon, 13 May 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b01366
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[ASAP] Cobalt-Catalyzed Diastereoselective Difluoroalkylation/Giese Addition Domino Reactions (Mon, 13 May 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b01400
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[ASAP] Total Synthesis and Stereochemical Confirmation of Heliolactone (Mon, 13 May 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b01402
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[ASAP] Radical Addition to <italic toggle="yes">N</italic>-Tosylimines via C–H Activation Induced by Decatungstate Photocatalyst (Mon, 13 May 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b01450
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[ASAP] Synthesis of a-Trifluoromethylamines by Cu-Catalyzed Regio- and Enantioselective Hydroamination of 1-Trifluoromethylalkenes (Mon, 13 May 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b01471
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[ASAP] Combining Bidentate Lewis Acid Catalysis and Photochemistry: Formal Insertion of <italic toggle="yes">o</italic>-Xylene into an Enamine Double Bond (Sun, 12 May 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b01020
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[ASAP] Cu-Catalyzed S<sub>N</sub>2' Substitution of Propargylic Phosphates with Vinylarene-Derived Chiral Nucleophiles: Synthesis of Chiral Allenes (Fri, 10 May 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b00908
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[ASAP] Synthesis of Bridged Biaryl Atropisomers via Sequential Cu- and Pd-Catalyzed Asymmetric Ring Opening and Cyclization (Fri, 10 May 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b01062
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[ASAP] Nickel-Catalyzed 1,2-Arylboration of Vinylarenes (Fri, 10 May 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b01120
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[ASAP] Mechanism of Brønsted-Base-Mediated Borylation of Propynols: A DFT Study (Fri, 10 May 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b01180
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[ASAP] External Reductant-Free Palladium-Catalyzed Reductive Insertion of Isocyanide: Synthesis of Polysubstituted Pyrroles and Its Applications as a Cysteine Probe (Fri, 10 May 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b01220
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[ASAP] Activation Relay on Rhodium-Catalyzed C–H Aminomethylation in Cooperation with Photoredox Catalysis (Fri, 10 May 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b01261
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[ASAP] Catalytic Selective Oxidative Coupling of Secondary <italic toggle="yes">N</italic>-Alkylanilines: An Approach to Azoxyarene (Thu, 09 May 2019)
TOC Graphic Organic Letters DOI: 10.1021/acs.orglett.9b01200
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