The Journal of Organic Chemistry



[ASAP] Visible-Light-Mediated Oxidative Coupling of Vinylarenes with Bromocarboxylates Leading to ?-Ketoesters (Fri, 15 Nov 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b02310
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[ASAP] Stereo- and Regiochemical Transannular Cyclization of a Common Hexahydro-1<italic toggle="yes">H</italic>-azonine to Afford Three Different Indolizidinone Dipeptide Mimetics (Fri, 15 Nov 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01861
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[ASAP] Synthesis of Functionalized 6,5- and 7,5-Azabicycloalkane Amino Acids by Metathesis Reactions (Fri, 15 Nov 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b02268
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[ASAP] Reductive Cleavage of Unactivated Carbon–Cyano Bonds under Ammonia-Free Birch Conditions (Fri, 15 Nov 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b02028
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[ASAP] Biomimetic Total Synthesis of <italic toggle="yes">Dysoxylum</italic> Alkaloids (Fri, 15 Nov 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b02093
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[ASAP] Synthesis of Sterically Congested 2,2'-Bi(Adamantyl)-Based Alcohol and Amines (Fri, 15 Nov 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b02293
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[ASAP] Palladium-Catalyzed [3+2] Annulation of Naphthalimide Acceptors and Thiophene Donors (Fri, 15 Nov 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b02372
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[ASAP] Mechanical Fixation by Porphyrin Connection: Synthesis and Transport Studies of a Bicyclic Dimer (Fri, 15 Nov 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b02327
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[ASAP] Cooperative Catalysis of Chiral Guanidine and Rh<sub>2</sub>(OAc)<sub>4</sub> in Asymmetric O–H Insertion of Carboxylic Acid: A Theoretical Investigation (Thu, 14 Nov 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.8b02850
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[ASAP] Correction to A Protonated Quinone Methide Stabilized by a Combination of Partial Aromatization and p-Interaction: Spectroscopic and Crystallographic Analysis (Thu, 14 Nov 2019)
The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b03002
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[ASAP] H-bonding vs Protonation of Alkynes in Regioselective Hydroamination Reactions: A Glimpse into the Reactivity of Arylogous Ynolethers and Ynamines (Thu, 14 Nov 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b02471
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[ASAP] Visible-Light-Catalyzed [3 + 1 + 2] Coupling Annulations for the Synthesis of Unsymmetrical Trisubstituted Amino-1,3,5-triazines (Thu, 14 Nov 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b02514
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[ASAP] Aromatic C–H Bond Functionalized via Zwitterion Intermediates to Construct Bioxindole Containing Continuous Quaternary Carbons (Thu, 14 Nov 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b02228
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[ASAP] Synthesis of Indolo- and Benzothieno[2,3-<italic toggle="yes">b</italic>]quinolines by a Cascade Cyclization of <italic toggle="yes">o</italic>-Alkynylisocyanobenzene Derivatives (Thu, 14 Nov 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b02081
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[ASAP] Three-Component Coupling of Aromatic Aldehydes, 1-Morpholino-2-nitroalkenes, and 3-Aminoazoles via Boron Trifluoride Etherate Catalysis: Reaction Pathway and Features of the Formation of Intermediates (Thu, 14 Nov 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b02286
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[ASAP] Base-Mediated Tunable Synthesis of 2-Trifluoromethylated Furans and Dihydrofuranols: Extraordinary Stable in Sulfuric Acid (Thu, 14 Nov 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b02326
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[ASAP] Tuning Isonitrile/Tetrazine Chemistry for Accelerated Deprotection and Formation of Stable Conjugates (Thu, 14 Nov 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b02522
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[ASAP] 1,1'-Biaceanthrylene and 2,2'-Biaceanthrylene: Models for Linking Larger Polycyclic Aromatic Hydrocarbons via Five-Membered Rings (Wed, 13 Nov 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b02118
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[ASAP] Hydrogen Abstraction from the C15 Position of the Cholesterol Skeleton (Wed, 13 Nov 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b02181
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[ASAP] Computationally Assisted Mechanistic Investigation into Hypervalent Iodine Catalysis: Cyclization of <italic toggle="yes">N</italic>-Allylbenzamide (Wed, 13 Nov 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b02623
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[ASAP] Solid-Phase Synthesis of Phosphate/Boranophosphate Chimeric DNAs Using the <italic toggle="yes">H</italic>-Phosphonate–<italic toggle="yes">H</italic>-Boranophosphonate Method (Wed, 13 Nov 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01257
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[ASAP] Correction to Fluorofunctionalization of C-C Bonds with Selectfluor: Synthesis of ß-Fluoropiperazines through a Substrate-Guided Reactivity Switch (Wed, 13 Nov 2019)
The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b02989
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[ASAP] Mechanism of Os-Catalyzed Oxidative Cyclization of 1,5-Dienes (Wed, 13 Nov 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b02174
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[ASAP] Rh(III)-Catalyzed C–H Activation/Cycloisomerization of <italic toggle="yes">N</italic>-Phenoxyacetamides with Enynones for One-Pot Assembly of Furylated 2-Alkenylphenols (Wed, 13 Nov 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b02534
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[ASAP] Synthesis of 5,12-Diazapentacenes and Their Properties (Wed, 13 Nov 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01628
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[ASAP] Synthesis of Heparan Sulfate- and Dermatan Sulfate-Related Oligosaccharides via Iterative Chemoselective Glycosylation Exploiting Conformationally Disarmed [2.2.2] <sc>l</sc>-Iduronic Lactone Thioglycosides (Wed, 13 Nov 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01594
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[ASAP] Introduction of Aryl Fluorosulfates into the Realm of Catellani Reaction Substrates (Tue, 12 Nov 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b02352
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[ASAP] Synthesis of <italic toggle="yes">N</italic>-Acyl Sulfamates from Fluorosulfonates and Potassium Trimethylsilyloxyl Imidates (Tue, 12 Nov 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b02394
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[ASAP] Methoxy Groups Increase Reactivity of Bifunctional Tetraarylphosphonium Salt Catalysts for Carbon Dioxide Fixation: A Mechanistic Study (Tue, 12 Nov 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b02581
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[ASAP] Copper-Catalyzed Cascade Denitrogenative Transannulation/Hydrolyzation of 3-Aminoindazoles toward 2,2-Disubstituted Indanones (Tue, 12 Nov 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b02303
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[ASAP] Synthesis of Fmoc-Protected Amino Alcohols via the Sharpless Asymmetric Aminohydroxylation Reaction Using FmocNHCl as the Nitrogen Source (Tue, 12 Nov 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b02491
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[ASAP] Synthesis of Butenolides via a Horner–Wadsworth–Emmons Cascading Dimerization Reaction (Tue, 12 Nov 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b02015
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[ASAP] Direct Transformation of N-Protected a,ß-Unsaturated ?-Amino Amides into ?-Lactams through a Base-Mediated Molecular Rearrangement (Mon, 11 Nov 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01936
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[ASAP] General Approach for the Liquid-Phase Fragment Synthesis of Orthogonally Protected Naturally Occurring Polyamines and Applications Thereof (Mon, 11 Nov 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b02066
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[ASAP] Donor–Acceptor p-Conjugated Enamines: Functional Group-Compatible Synthesis from Amides and Their Photoabsorption and Photoluminescence Properties (Mon, 11 Nov 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b02267
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[ASAP] I<sub>2</sub>–DMSO–H<sub>2</sub>O: A Metal-Free Combination System for the Oxidative Addition of Alkynes to Access (<italic toggle="yes">E</italic>)-a-Iodo-ß-methylsulfonylalkenes (Mon, 11 Nov 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b02302
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[ASAP] Characterizing Cation Chemistry for Anion Exchange Membranes—A Product Study of Benzylimidazolium Salt Decompositions in the Base (Mon, 11 Nov 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b02493
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[ASAP] Enantioselective Synthesis of CF<sub>3</sub>S-Containing Compounds via Ir-Catalyzed Allylic Alkylations of CF<sub>3</sub>S-Substituted Functionalized Methylene Derivatives (Mon, 11 Nov 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b02123
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[ASAP] Mn-Enabled Radical-Based Alkyl–Alkyl Cross-Coupling Reaction from 4-Alkyl-1,4-dihydropyridines (Mon, 11 Nov 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b02323
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[ASAP] Development of Triazinone-Based Condensing Reagents for Amide Formation (Fri, 08 Nov 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01261
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[ASAP] Peptoid Helix Displaying Flavone and Porphyrin: Synthesis and Intramolecular Energy Transfer (Fri, 08 Nov 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b02358
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[ASAP] Synthesis of Enantiopure e-Oxapipecolic Acid (Fri, 08 Nov 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b02382
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[ASAP] Double <italic toggle="yes">ortho</italic>-C–H Activation/Annulation of Benzamides with Aryl Alkynes: A Route to Double-Helical Polycyclic Heteroaromatics (Fri, 08 Nov 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b02339
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[ASAP] Stereocontrolled Total Synthesis of (+)-Isolaurenidificin and (-)-Bromlaurenidificin (Fri, 08 Nov 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b02532
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[ASAP] Regioselective Synthesis of Functionalized 3- or 5-Fluoroalkyl Isoxazoles and Pyrazoles from Fluoroalkyl Ynones and Binucleophiles (Fri, 08 Nov 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b02258
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[ASAP] Chiral-at-Metal Rh(III) Complex Catalyzed Cascade Reduction-Michael Addition Reaction (Fri, 08 Nov 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b02243
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[ASAP] Unexpected Synthesis, Properties, and Nonvolatile Memory Device Application of Imidazole-Fused Azaacenes (Thu, 07 Nov 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b02156
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[ASAP] <italic toggle="yes">De Novo</italic> Asymmetric Synthesis of Avocadyne, Avocadene, and Avocadane Stereoisomers (Thu, 07 Nov 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b02391
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[ASAP] One-Pot Synthesis of <italic toggle="yes">Aza</italic>-Morita-Baylis-Hillman Adducts via Zinc-Mediated Allylation of 4-Bromocrotonates and Imines (Thu, 07 Nov 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b02434
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[ASAP] Difluoromethylation of Phenols and Thiophenols with the <italic toggle="yes">S</italic>-(Difluo-romethyl)sulfonium Salt: Reaction, Scope, and Mechanistic Study (Thu, 07 Nov 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b02424
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