The Journal of Organic Chemistry



[ASAP] Enantio- and Diastereoselective Two-Pot Synthesis of Isoquinuclidines from Glutaraldehyde and <italic toggle="yes">N</italic>-Aryl Imines with DFT Calculations (Tue, 17 Sep 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01865
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[ASAP] Divergent Synthesis of Methylene Lactone- and Methylene Lactam-Based Spiro Compounds: Utility of Amido-Functionalized ?-Hydroxylactam as a Precursor for Cytotoxic <italic toggle="yes">N</italic>,<italic toggle="yes">O</italic>- and <italic toggle="yes">N</italic>,<italic toggle="yes">N</italic>-Spiro Compounds (Tue, 17 Sep 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b02038
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[ASAP] <italic toggle="yes">N-</italic>Morpholinomethyl-5-lithiotetrazole: A Reagent for the One-Pot Synthesis of 5-(1-Hydroxyalkyl)tetrazoles (Tue, 17 Sep 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01885
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[ASAP] Cobalt-Catalyzed Carbonylative Synthesis of Phthalimides from <italic toggle="yes">N</italic>-(Pyridin-2-ylmethyl)benzamides with TFBen as the CO Source (Mon, 16 Sep 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01890
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[ASAP] Synthetic Studies toward the Total Synthesis of Tautomycetin (Mon, 16 Sep 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01712
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[ASAP] Fenton-Inspired C–H Functionalization: Peroxide-Directed C–H Thioetherification (Mon, 16 Sep 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01979
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[ASAP] Visible Light-Induced Co- or Cu-Catalyzed Selenosulfonylation of Alkynes: Synthesis of ß-(Seleno)vinyl Sulfones (Mon, 16 Sep 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01626
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[ASAP] DFT Studies on Metal-Controlled Regioselective Amination of <italic toggle="yes">N</italic>-Acylpyrazoles with Azodicarboxylates (Fri, 13 Sep 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01863
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[ASAP] Radical-Stimulated Nucleophile Release (Fri, 13 Sep 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b02159
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[ASAP] Synthetic Methodologies for Perfluoroaryl-Substituted (Diaryl)methylphosphonates, -Phosphinates via S<sub>N</sub>Ar Reaction (Fri, 13 Sep 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01402
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[ASAP] Transacylation in Ferrocenoyl-Purines. NMR and Computational Study of the Isomerization Mechanism (Thu, 12 Sep 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01944
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[ASAP] Donor–Acceptor–Donor NIR II Emissive Rhodindolizine Dye Synthesized by C–H Bond Functionalization (Thu, 12 Sep 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01860
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[ASAP] Direct C–H Methylsulfonylation of Alkenes with the Insertion of Sulfur Dioxide (Thu, 12 Sep 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01729
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[ASAP] Development of an Imine Chaperone for Selective C–H Functionalization of Alcohols via Radical Relay (Thu, 12 Sep 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b02052
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[ASAP] Enantiospecific Entry to a Common Decalin Intermediate for the Syntheses of Highly Oxygenated Terpenoids (Wed, 11 Sep 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01937
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[ASAP] Synthesis and Reactivity of 5-Heterotruxenes Containing Sulfur or Nitrogen as the Heteroatom (Wed, 11 Sep 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01397
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[ASAP] Synthesis of Central Chirality-Containing Triarylmethanols and Triarylmethyl Radicals with Extraordinarily Stable Configurations (Wed, 11 Sep 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01675
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[ASAP] Protecting-Group-Free Total Synthesis of Chatenaytrienin-2 (Wed, 11 Sep 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01952
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[ASAP] Copper-Catalyzed Regioselective sp<sup>3</sup> C–H Azidation of Alkyl Substituents of Indoles and Tetrahydrocarbazoles (Wed, 11 Sep 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01742
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[ASAP] Gold-Catalyzed Synthesis of 6-Hydroxyindoles from Alkynylcyclohexadienones and Substituted Amines (Wed, 11 Sep 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b02023
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[ASAP] N-Heterocyclic Carbene Ligand-Controlled Chemodivergent Suzuki–Miyaura Cross Coupling (Wed, 11 Sep 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01692
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[ASAP] Formation of Enol Ethers by Radical Decarboxylation of a-Alkoxy ß-Phenylthio Acids (Wed, 11 Sep 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b02042
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[ASAP] Hunterines A–C, Three Unusual Monoterpenoid Indole Alkaloids from <italic toggle="yes">Hunteria zeylanica</italic> (Tue, 10 Sep 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01835
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[ASAP] Protocols for the Syntheses of 2,2'-Bis(indolyl)arylmethanes, 2-Benzylated Indoles, and 5,7-Dihydroindolo[2,3-<italic toggle="yes">b</italic>]carbazoles (Tue, 10 Sep 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b02124
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[ASAP] Forging C–S Bonds through Nickel-Catalyzed Aryl Anhydrides with Thiophenols: Decarbonylation or Decarbonylation Accompanied by Decarboxylation (Tue, 10 Sep 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01746
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[ASAP] Studies on Long-Lived (Pentafluorosulfanyl)phenyl-Substituted Carbocations (Tue, 10 Sep 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01622
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[ASAP] Electron Push–Pull Effects in 3,9-Bis(<italic toggle="yes">p</italic>-(R)-diphenylamino)perylene and Constraint on Emission Color Tuning (Tue, 10 Sep 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01849
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[ASAP] <italic toggle="yes">N</italic>-Aminopyridinium Ylide-Directed, Copper-Promoted Amination of sp<sup>2</sup> C–H Bonds (Tue, 10 Sep 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01847
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[ASAP] Unexpected Rearrangement of Dilithiated Isoindoline-1,3-diols into 3-Aminoindan-1-ones via <italic toggle="yes">N</italic>-Lithioaminoarylcarbenes: A Combined Synthetic and Computational Study (Tue, 10 Sep 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01217
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[ASAP] C–N Coupling via Antiaromatic Endocyclic Nitrenium Ions (Tue, 10 Sep 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01921
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[ASAP] Direct C–H Bond Imidation with Benzoyl Peroxide as a Mild Oxidant and a Reagent (Tue, 10 Sep 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01765
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[ASAP] Catalytic Asymmetric Synthesis of Diketopiperazines by Intramolecular Tsuji–Trost Allylation (Tue, 10 Sep 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01994
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[ASAP] Palladium-Catalyzed Coupling of Terminal Alkynes with Benzyl Ammonium Salts (Tue, 10 Sep 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01877
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[ASAP] Multicomponent Tether Catalysis Synthesis of Highly Functionalized 4-(Pyridin-2-ylmethyl)-2-aminopyrroles via Cascade Reaction Is Accompanied by Decarboxylation (Mon, 09 Sep 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01814
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[ASAP] Asymmetric Palladium-Catalyzed C–H Functionalization Cascade for Synthesis of Chiral 3,4-Dihydroisoquinolones (Mon, 09 Sep 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01372
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[ASAP] Metal-Free Transamidation of Secondary Amides by N–C Cleavage (Mon, 09 Sep 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b02013
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[ASAP] Cu(I)-Catalyzed Asymmetric Mannich Reaction of Glycine Schiff Bases to Ketimines (Mon, 09 Sep 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01566
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[ASAP] Redox Property of Enamines (Mon, 09 Sep 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b02003
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[ASAP] Synthesis of 2-Amino-5-acylthiazoles by a Tertiary Amine-Promoted One-Pot Three-Component Cascade Cyclization Using Elemental Sulfur as a Sulfur Source (Mon, 09 Sep 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b02032
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[ASAP] Lewis Base-Catalyzed Enantioselective Conjugate Reduction of ß,ß-Disubstituted a,ß-Unsaturated Ketones with Trichlorosilane: <italic toggle="yes">E</italic>/<italic toggle="yes">Z</italic>-Isomerization, Regioselectivity, and Synthetic Applications (Mon, 09 Sep 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01298
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[ASAP] Total Synthesis of Phenanthroquinolizidine Alkaloids Using a Building Block Strategy (Mon, 09 Sep 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01768
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[ASAP] Regio- and Stereoselective Carboindation of Internal Alkynyl Ethers with Organosilicon or -stannane Nucleophiles (Mon, 09 Sep 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01505
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[ASAP] Palladium-Catalyzed Cascade Annulation/Allylation of Alkynyl Oxime Ethers with Allyl Halides: Rapid Access to Fully Substituted Isoxazoles (Mon, 09 Sep 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01593
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[ASAP] Redox-Neutral Rhodium(III)-Catalyzed Annulation of Arylhydrazines with Sulfoxonium Ylides To Synthesize 2-Arylindoles (Fri, 06 Sep 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01815
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[ASAP] Total Synthesis of A54145 Factor D (Fri, 06 Sep 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01938
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[ASAP] Liquid-Phase Hydrogenation of Nitriles to Amines Facilitated by a Co(II)/Zn(0) Pair: A Ligand-Free Catalytic Protocol (Fri, 06 Sep 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01544
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[ASAP] Rh(II)-Catalyzed Denitrogenative Transannulation of <italic toggle="yes">N</italic>-Sulfonyl-1,2,3-triazolyl Cyclohexadienones for the Synthesis of Benzofurans and Cyclopropa[<italic toggle="yes">cd</italic>]indole-carbaldehydes (Fri, 06 Sep 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01924
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[ASAP] Identifying Amidyl Radicals for Intermolecular C–H Functionalizations (Fri, 06 Sep 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01774
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[ASAP] Threading of Conformationally Stable Calix[6]arene Wheels Substituted at the Methylene Bridges (Fri, 06 Sep 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01779
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[ASAP] Kinetic Stabilization of Carbazole Nitroxides by Inclusion in a Macrocage and Their Electron Spin Resonance Characterization (Fri, 06 Sep 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01686
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