The Journal of Organic Chemistry

The Palladium-Catalyzed Intramolecular Alder-Ene Reactions of O- and N-Linked 1,6-Enynes Incorporating Triethylsilyl Capping Groups (Tue, 14 Nov 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02355
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Bimetallic Cobalt–Rhodium Nanoparticle-Catalyzed Reductive Amination of Aldehydes with Nitroarenes Under Atmospheric Hydrogen (Tue, 14 Nov 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02019
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Ring-Fused Cyclic Aminals from Tetrahydro-β-carboline-Based Dipeptide Compounds (Tue, 14 Nov 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01656
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Rh(III)-Catalyzed Direct ortho-Chalcogenation of Phenols and Anilines (Tue, 14 Nov 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02221
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“On Water” Direct C-3 Arylation of 2H-Pyrazolo[3,4-b]pyridines (Mon, 13 Nov 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02136
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Intramolecular Diels–Alder Reactions of Tethered Enoate Substituted Furans Induced by Dialkylaluminum Chloride (Mon, 13 Nov 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02117
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Synthesis of Chiral Tritylpyrrolidine Derivatives and Their Application to Asymmetric Benzoyloxylation (Mon, 13 Nov 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02562
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Short Enantioselective Total Syntheses of Cheloviolenes A and B and Dendrillolide C via Convergent Fragment Coupling Using a Tertiary Carbon Radical (Mon, 13 Nov 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02458
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Spiropiperidine Sultam and Lactam Templates: Diastereoselective Overman Rearrangement and Metathesis followed by NH Arylation (Mon, 13 Nov 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02096
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Observation of a Tricyclic[4.1.0.02,4]heptane During a Michael Addition-Ring Closure Reaction and a Computational Study on Its Mechanism of Formation (Fri, 10 Nov 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02218
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Enantioselective Synthesis of Alkylthioetherpyrrolidine Derivatives via [3+2] Cycloaddition of α-Thioacrylates with Isocyanoacetates (Fri, 10 Nov 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02266
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Theoretical Elucidation of the Mechanism and Kinetic Experimental Phenomena on the Esterification of α-Tocopherol with Succinic Anhydride: Catalysis of a Histidine Derivative vs an Imidazolium-Based Ionic Liquid (Fri, 10 Nov 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02102
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Hydroxy-Assisted Regio- and Stereoselective Synthesis of Functionalized 4-Methylenepyrrolidine Derivatives via Phosphine-Catalyzed [3 + 2] Cycloaddition of Allenoates with o-Hydroxyaryl Azomethine Ylides (Fri, 10 Nov 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02560
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Lewis Acid Triggered Vinylcyclopropane–Cyclopentene Rearrangement (Fri, 10 Nov 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02351
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Synthesis of 2-Aryl-3-sulfonylchromans via Knoevenagel Condensation and Reduction Protocol (Thu, 09 Nov 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02392
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Organocatalytic and Late-Stage CH-Functionalization Enabled Asymmetric Synthesis of Communesin F and Putative Communesins (Thu, 09 Nov 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02426
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Synthesis of Polysubstituted Pyrroles through a Formal [4 + 1] Cycloaddition/E1cb Elimination/Aromatization Sequence of Sulfur Ylides and α,β-Unsaturated Imines (Thu, 09 Nov 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01931
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Phellilane L, Sesquiterpene Metabolite of Phellinus linteus: Isolation, Structure Elucidation, and Asymmetric Total Synthesis (Thu, 09 Nov 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02141
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Friedel–Crafts Acylation Reactions of BN-Substituted Arenes (Thu, 09 Nov 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02343
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Total Synthesis of Kanamienamide and Clarification of Biological Activity (Wed, 08 Nov 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02288
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Synthesis and Optical Properties of Excited-State Intramolecular Proton Transfer Active π-Conjugated Benzimidazole Compounds: Influence of Structural Rigidification by Ring Fusion (Wed, 08 Nov 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01967
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Palladium-Catalyzed Construction of Tetracyclic Scaffolds via the 1,7-Enyne Carbocyclization/Iodophenol Dearomatization Cascade (Wed, 08 Nov 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02196
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Copper-Catalyzed Azidative Multifunctionalization of Alkynes (Wed, 08 Nov 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02148
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Support for a Dioxyallyl Cation in the Mechanism Leading to (−)-Levoglucosenone (Wed, 08 Nov 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02109
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Straightforward S–S Bond Formation via the Oxidation of S-Acetyl by Iodine in the Presence of N-Iodosuccinimide (Tue, 07 Nov 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02367
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Organocatalytic Asymmetric Allylic Alkylation of Morita–Baylis–Hillman Carbonates with Diethyl 2-Aminomalonate Assisted by In Situ Protection (Tue, 07 Nov 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02064
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Scaling the Amphiphilic Character and Antimicrobial Activity of Gramicidin S by Dihydroxylation or Ketal Formation (Tue, 07 Nov 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02177
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Organocatalytic Enantioselective Michael–Acetalization–Henry Reaction Cascade of 2-Hydroxynitrostyrene and 5-Oxohexanal for the Entry to the Hexahydro-6H-benzo[c]chromenones with Four Consecutive Stereogenic Centers and an Approach to Aflatoxin Analogues (Tue, 07 Nov 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02178
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Nucleophilic Addition of Ketones To Acetylenes and Allenes: A Quantum-Chemical Insight (Tue, 07 Nov 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02263
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Diastereoselective Synthesis of Functionalized Diketopiperazines through Post-transformational Reactions (Tue, 07 Nov 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01855
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Rhodium-Catalyzed sp2 C–H Acetoxylation of N-Aryl Azaindoles/N-Heteroaryl Indolines (Tue, 07 Nov 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02203
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Application of the EF and GH Fragments to the Synthesis of Idraparinux (Tue, 07 Nov 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02497
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Camphorsulfonic Acid Catalyzed One-Pot Three-Component Reaction for the Synthesis of Fused Quinoline and Benzoquinoline Derivatives (Tue, 07 Nov 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02159
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Enantiospecific Semisynthesis of Puupehedione-Type Marine Natural Products (Tue, 07 Nov 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02413
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Synthesis of Allahabadolactone A (Tue, 07 Nov 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02368
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General and Catalytic Enantioselective Approach to Isopavine Alkaloids (Tue, 07 Nov 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02385
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Iron Catalyzed Hydroboration of Aldehydes and Ketones (Tue, 07 Nov 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02020
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Chemoselective α-Methylenation of Aromatic Ketones Using the NaAuCl4/Selectfluor/DMSO System (Tue, 07 Nov 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01790
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Total Synthesis and Biological Mode of Action of WAP-8294A2: A Menaquinone-Targeting Antibiotic (Tue, 07 Nov 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02318
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Application of Vinyl Azides in Chemical Synthesis: A Recent Update (Fri, 03 Nov 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02455
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Molecular Spur Gears Based on a Switchable Quinquepyridine Foldamer Acting as a Stator (Fri, 03 Nov 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01864
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Isothiocyanyl Alanine as a Synthetic Intermediate for the Synthesis of Thioureayl Alanines and Subsequent Aminotetrazolyl Alanines (Fri, 03 Nov 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02103
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Palladium-Catalyzed Diastereoselective Synthesis of 3-Arylbutanoic Acid Derivatives (Thu, 02 Nov 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02104
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Reductive Alkylation of Tertiary Lactams via Addition of Organocopper (RCu) Reagents to Thioiminium Ions (Thu, 02 Nov 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02150
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Oxidant and Transition-Metal-Free Photoinduced Direct Oxidative Annulation of 1-Aryl-2-(furan/thiophen-2-yl)butane-1,3-diones (Thu, 02 Nov 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01839
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Protecting-Group-Free Synthesis of 1-Phenylisoquinolin-4-ols: Thermal Cyclization of Methyl 2-[(Diphenylmethylidene)amino]acetates (Thu, 02 Nov 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02240
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Tunable Heck–Mizoroki Reaction of Dibromonaphthalene Diimide with Aryl Ethylenes: Design, Synthesis, and Characterization of Coplanar NDI-Based Conjugated Molecules (Thu, 02 Nov 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02140
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Stereochemistry of Nucleophilic Substitutions on Benzyl-silane and -germane Cation Radicals: Application of the Endocyclic Restriction Test (Thu, 02 Nov 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01892
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Cyclobutyl-Containing Rigid Analogues of Threonine: Synthesis and Physical Chemical Properties (Thu, 02 Nov 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02259
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N-Heterocycle-Forming Amino/Carboperfluoroalkylations of Aminoalkenes by Using Perfluoro Acid Anhydrides: Mechanistic Studies and Applications Directed Toward Perfluoroalkylated Compound Libraries (Wed, 01 Nov 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02307
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Ru/Cu Photoredox or Cu/Ag Catalyzed C4–H Sulfonylation of 1-Naphthylamides at Room Temperature (Wed, 01 Nov 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01917
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Correction to “Diverting Reactive Intermediates Toward Unusual Chemistry: Unexpected Anthranil Products from Davis–Beirut Reaction” (Wed, 01 Nov 2017)
The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02695
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Reinvestigation of the Substitutions Reaction of Stereogenic Phosphoryl Compounds: Stereochemistry, Mechanism, and Applications (Wed, 01 Nov 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01326
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Asymmetric Syntheses of 3-Deoxy-3-aminosphingoid Bases: Approaches Based on Parallel Kinetic Resolution and Double Asymmetric Induction (Wed, 01 Nov 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02233
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Nonstabilized Azomethine Ylides in the Mannich Reaction: Synthesis of 3,3-Disubstituted Pyrrolidines, Including Oxindole Alkaloids (Wed, 01 Nov 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02193
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Protocol for the Direct Conversion of Lactones to Lactams Mediated by 1,5,7-Triazabicyclo[4.4.0]dec-5-ene: Synthesis of Pyridopyrazine-1,6-diones (Wed, 01 Nov 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02079
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Triplet Sensitized Photodenitrogenation of Δ2-1,2,3-Triazolines To Form Aziridines in Solution and in the Crystalline State: Observation of the Triplet 1,3-Alkyl-aminyl Biradical (Wed, 01 Nov 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01924
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Synthesis of Furo[2,3-c]pyridazines via Tandem Transition-Metal Catalysis (Tue, 31 Oct 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01819
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Reversible Redox Switching of Chromophoric Phenylmethylenepyrans by Carbon–Carbon Bond Making/Breaking (Tue, 31 Oct 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02199
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Conversion of Alcohols to Phosphorothiolates Using a Thioiminium Salt as Coupling Agent (Tue, 31 Oct 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01657
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Asymmetric Darzens Reaction of Isatins with Diazoacetamides Catalyzed by Chiral BINOL–Titanium Complex (Tue, 31 Oct 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02439
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Infrared Fingerprints of nN → σ*NH Hyperconjugation in Hydrazides (Tue, 31 Oct 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01985
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Synthesis of 5′-Thio-3′-O-ribonucleoside Phosphoramidites (Tue, 31 Oct 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01484
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Photoredox-Catalyzed Deoxygenative Intramolecular Acylation of Biarylcarboxylic Acids: Access to Fluorenones (Tue, 31 Oct 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02197
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Why Do Cumulene Ketones Kink? (Mon, 30 Oct 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02089
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Synthesis of Enantiopure Mixed Alkyl-Aryl Vicinal Diamines by the Diaza-Cope Rearrangement: A Synthesis of (+)-CP-99,994 (Mon, 30 Oct 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01751
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A Quantitative Analysis of Factors Influencing Ease of Formation and σ-Bonding Strength of Oxa- and Thia-N-Heterocyclic Carbenes (Mon, 30 Oct 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02283
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Strain-Promoted Nitration of 3-Cyclopropylideneprop-2-en-1-ones and the Application for the Synthesis of Pyrroles (Mon, 30 Oct 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02087
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Structure-Based Kinetic Control in a Domino Process: A Powerful Tool Toward Molecular Diversity in Chromone Series (Mon, 30 Oct 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01996
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Molecular Engineering of Near Infrared Absorbing Thienopyrazine Double Donor Double Acceptor Organic Dyes for Dye-Sensitized Solar Cells (Mon, 30 Oct 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01750
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Palladium(0)-Catalyzed Carbonylative One-Pot Synthesis of N-Acylguanidines (Fri, 27 Oct 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02294
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Three-Step Synthesis of Chiral Spirocyclic Oxaphospholenes (Fri, 27 Oct 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02227
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Asymmetric α-Allylation of α-Substituted β-Ketoesters with Allyl Alcohols (Fri, 27 Oct 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02188
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Total Synthesis of Glycinocins A–C (Fri, 27 Oct 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01959
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Synthesis of a Pentasaccharide Fragment Related to the Inner Core Region of Rhizobial and Agrobacterial Lipopolysaccharides (Thu, 26 Oct 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02172
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Diastereoselective Desymmetrization of Prochiral Cyclopentenediones via Cycloaddition Reaction with N-Phenacylbenzothiazolium Bromides (Thu, 26 Oct 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01964
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Correction to Origins of Regioselectivity in the Fischer Indole Synthesis of a Selective Androgen Receptor Modulator (Thu, 26 Oct 2017)
The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02416
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TBHP/TBAI-Mediated Oxidative Cascade Reaction Consisting of Dimerization, Cyclization, and 1,2-Aryl Migration: Metal-Free Synthesis of Pyrrolin-4-ones and Highly Substituted Pyrroles (Thu, 26 Oct 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02491
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Microwave Synthesis of Thionated Naphthalene Diimide-Based Small Molecules and Polymers (Thu, 26 Oct 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02162
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Transition-Metal-Free [3+2] Cycloaddition of Dehydroaminophosphonates and N-Tosylhydrazones: Access to Aminocyclopropanephosphonates with Adjacent Quaternary-Tetrasubstituted Carbon Centers (Thu, 26 Oct 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01862
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Synthesis of Stable [28π] m-Benzihexaphyrins (1.0.0.1.1.1) (Thu, 26 Oct 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02095
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Synthesis of Quaternary-Substituted Thiazolines via Halocyclization of S-Allyl Thioimidate Salts (Tue, 24 Oct 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02299
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The Difference a Single Atom Can Make: Synthesis and Design at the Chemistry–Biology Interface (Fri, 13 Oct 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b02088
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Structural Revision of Baulamycin A and Structure–Activity Relationships of Baulamycin A Derivatives (Mon, 02 Oct 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01719
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