The Journal of Organic Chemistry



[ASAP] Inhibitory Evaluation of aPMM/PGM from <italic toggle="yes">Pseudomonas aeruginosa</italic>: Chemical Synthesis, Enzyme Kinetics, and Protein Crystallographic Study (Tue, 16 Jul 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01305
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[ASAP] Transition-Metal-Free Synthesis of Fused Quinazolinones by Oxidative Cyclization of <italic toggle="yes">N</italic>-Pyridylindoles (Tue, 16 Jul 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01170
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[ASAP] Synthesis of ?-Pyrones from Formal [4 + 2] Cyclization of Ketene Dithioacetals with Acyl Chlorides (Tue, 16 Jul 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01254
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[ASAP] Nickel-Catalyzed Direct Alkenylation of Methyl Heteroarenes with Primary Alcohols (Tue, 16 Jul 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01517
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[ASAP] A Photochemical Route to Optically Active Hexahydro-4<italic toggle="yes">H</italic>-furopyranol, a High-Affinity P2 Ligand for HIV-1 Protease Inhibitors (Tue, 16 Jul 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01361
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[ASAP] Cyanoacetylenes as Triggers and Partners in KOH-Assisted Assemblies of Quinoline-Based Dihydropyrimido[1,2-<italic toggle="yes">a</italic>]quinolin-3-ones on Water (Tue, 16 Jul 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01482
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[ASAP] Palladium-Catalyzed <italic toggle="yes">ortho</italic>-C–H Methylation of Benzoic Acids (Mon, 15 Jul 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01204
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[ASAP] Rh(III)-Catalyzed C(8)–H Activation of Quinoline <italic toggle="yes">N</italic>-Oxides: Regioselective C–Br and C–N Bond Formation (Fri, 12 Jul 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01538
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[ASAP] [3 + 2]-Cycloaddition of Azaoxyallyl Cations with 1,2-Benzisoxazoles: A Rapid Entry to Oxazolines (Fri, 12 Jul 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01166
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[ASAP] General Approach To Construct Azepino[2,3-<italic toggle="yes">b</italic>:4,5-<italic toggle="yes">b</italic>']diindoles, Azocino[2,3-<italic toggle="yes">b</italic>:4,5-<italic toggle="yes">b</italic>']diindoles, and Azonino[2,3-<italic toggle="yes">b</italic>:4,5-<italic toggle="yes">b</italic>']diindoles via Rh(II)-Catalyzed Reactions of 3-Diazoindolin-2-imines with 3-(Bromoalkyl)indoles (Fri, 12 Jul 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01169
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[ASAP] Synthesis of Diiodinated All-Carbon 3,3'-Diphenyl-1,1'-spirobiindene Derivatives via Cascade Enyne Cyclization and Electrophilic Aromatic Substitution (Thu, 11 Jul 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01418
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[ASAP] Switchable Synthesis of Arylalkynes and Phthalides via Controllable Palladium-Catalyzed Alkynylation and Alkynylation–Annulation of Benzoic Acids with Bromoalkynes (Thu, 11 Jul 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01102
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[ASAP] Meso-Fused Carbatriphyrins(2.1.1) and Its Organo Phosphorus(V) Complex (Thu, 11 Jul 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01015
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[ASAP] Correction to Simple Chiral Derivatization Protocols for <sup>1</sup>H NMR and <sup>19</sup>F NMR Spectroscopic Analysis of the Enantiopurity of Chiral Diols (Thu, 11 Jul 2019)
The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01735
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[ASAP] Theoretical Insight into the Mechanism and Origin of Divergent Reactivity in the Synthesis of Benzo-Heterocycles from <italic toggle="yes">o</italic>-Alkynylbenzamides Catalyzed by Gold and Platinum Complexes (Thu, 11 Jul 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01441
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[ASAP] Preparation and Application of Amino Phosphine Ligands Bearing Spiro[indane-1,2'-pyrrolidine] Backbone (Thu, 11 Jul 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b00875
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[ASAP] Formation and Reactivity of Triplet Vinylnitrenes as a Function of Ring Size (Thu, 11 Jul 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01191
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[ASAP] Sulfur-Mediated Allylic C–H Arylation, Epoxidation, and Aziridination (Thu, 11 Jul 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01438
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[ASAP] Fluorium-Initiated Dealkylative Cyanation of Thioethers to Thiocyanates (Wed, 10 Jul 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b00965
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[ASAP] [4 + 2]-Annulation of MBH-Acetates of Acetylenic Aldehydes with Imidazoles/Benzimidazoles To Access Imidazo[1,2-<italic toggle="yes">a</italic>]pyridines/Benzimidazo[1,2-<italic toggle="yes">a</italic>]pyridines (Wed, 10 Jul 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01118
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[ASAP] Double Addition of Alkynyllithium Reagents to Amides/Lactams: A Direct and Flexible Synthesis of 3-Amino-1,4-diynes Bearing an Aza-Quaternary Carbon Center (Tue, 09 Jul 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01416
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[ASAP] Designing of Push–Pull Chromophores with Tunable Electronic and Luminescent Properties Using Urea as the Electron Donor (Mon, 08 Jul 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b00841
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[ASAP] Photoactive Boron–Nitrogen–Carbon Hybrids: From Azo-borazines to Polymeric Materials (Mon, 08 Jul 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01046
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[ASAP] Diastereoselective Construction of 2-Aminoindanones via an In(OTf)<sub>3</sub>-Catalyzed Domino Reaction (Mon, 08 Jul 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b00876
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[ASAP] Manganese-Catalyzed and Mediated Synthesis of Arylphosphinates and Related Compounds (Mon, 08 Jul 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01239
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[ASAP] Dehydrogenation of Alcohols to Carboxylic Acid Catalyzed by in Situ-Generated Facial Ruthenium-<bold>CPP</bold> Complex (Fri, 05 Jul 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01100
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[ASAP] Lewis Acid-Catalyzed Intermolecular Annulation: Three-Component Reaction toward Imidazo[1,2-<italic toggle="yes">a</italic>]pyridine Thiones (Fri, 05 Jul 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01188
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[ASAP] Sekgranaticin, a SEK34b-Granaticin Hybrid Polyketide from <italic toggle="yes">Streptomyces</italic> sp. 166# (Fri, 05 Jul 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01022
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[ASAP] 2<italic toggle="yes">H</italic>-Indazole Tautomers Stabilized by Intra- and Intermolecular Hydrogen Bonds (Fri, 05 Jul 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01021
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[ASAP] Synthesis of Cryptophane-223-Type Derivatives with Dual Functionalization (Fri, 05 Jul 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01093
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[ASAP] Copper-Catalyzed Anomeric O-Arylation of Carbohydrate Derivatives at Room Temperature (Fri, 05 Jul 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01218
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[ASAP] Cp*Ir(III)-Catalyzed C–H/O–H Functionalization of Salicylaldehydes for the Synthesis of Chromones at Room Temperature (Fri, 05 Jul 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01139
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[ASAP] Synthesis of D–A–A and D–A–D Pyrimidine p-Systems Using Triorganoindium Reagents: Optical, Vibrational, and Electrochemical Studies (Fri, 05 Jul 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b00643
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[ASAP] Synthesis of the Methyl Analog of 2'-<italic toggle="yes">O</italic>,4'-<italic toggle="yes">C</italic>-Ethylene-Bridged 5-Methyluridine via Intramolecular Radical Cyclization and Properties of Modified Oligonucleotides (Fri, 05 Jul 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01035
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[ASAP] Stereoselective Assembly of Multifunctional Spirocyclohexene Pyrazolones That Induce Autophagy-Dependent Apoptosis in Colorectal Cancer Cells (Wed, 03 Jul 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01098
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[ASAP] Annulation of Benzamides with Arynes Using Palladium with Photoredox Dual Catalysis (Tue, 02 Jul 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b00893
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[ASAP] Palladium-Catalyzed Cross-Coupling of 2-Iodoglycals with <italic toggle="yes">N</italic>-Tosylhydrazones: Access to 2-C-Branched Glycoconjugates and Oxadecalins (Tue, 02 Jul 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01056
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[ASAP] Synthesis of 4,4-Difluoroalkenes by Coupling of a-Substituted a,a-Difluoromethyl Halides with Allyl Sulfones under Photoredox Catalyzed Conditions (Tue, 02 Jul 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b00901
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[ASAP] Second-Generation Synthesis of the Northern Fragment of Mandelalide A: Role of p-Stacking on Sharpless Dihydroxylation of <italic toggle="yes">cis</italic>-Enynes (Tue, 02 Jul 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01153
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[ASAP] Two-Step Transformation of Aliphatic Polyketones into p-Conjugated Polyimines (Tue, 02 Jul 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01119
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[ASAP] Diverse Chemosensitizing 8,9-Secolindenane-Type Sesquiterpenoid Oligomers and Monomers from <italic toggle="yes">Sarcandra glabra</italic> (Tue, 02 Jul 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b00986
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[ASAP] Aryl Carbamates: Mechanisms of Orthosodiations and Snieckus–Fries Rearrangements (Mon, 01 Jul 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b00968
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[ASAP] Synthesis of <italic toggle="yes">N</italic>-Pyrrolyl(furanyl)-Substituted Piperazines, 1,4-Dizepanes, and 1,4-Diazocanes (Mon, 01 Jul 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b00867
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[ASAP] The Synthesis of Bicyclo[4.2.1]nona-2,4,7-trienes by [6p + 2p]-Cycloaddition of 1-Substituted 1,3,5-Cycloheptatrienes Catalyzed by Titanium and Cobalt Complexes (Mon, 01 Jul 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b00996
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[ASAP] Photoredox-Catalyzed Radical Cascade Reaction To Synthesize Fluorinated Pyrrolo[1,2-<italic toggle="yes">d</italic>]benzodiazepine Derivatives (Mon, 01 Jul 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b00937
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[ASAP] Visible-Light-Triggered Selective Intermolecular [2+2] Cycloaddition of Extended Enones: 2-Oxo-3-enoates and 2,4-Dien-1-ones with Olefins (Mon, 01 Jul 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01273
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[ASAP] Lactam Hydrogen Bonds as Control Elements in Enantioselective Transition-Metal-Catalyzed and Photochemical Reactions (Sun, 30 Jun 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b01299
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[ASAP] Visible Light-Mediated [2 + 2] Cycloaddition Reactions of 1,4-Quinones and Terminal Alkynes (Fri, 28 Jun 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b00855
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[ASAP] Synthesis of Fullerene–Fluorene Dyads through the Platinum-Catalyzed Reactions of [60]Fullerene with 9-Ethynyl-9<italic toggle="yes">H</italic>-fluoren-9-yl Carboxylates (Fri, 28 Jun 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b00932
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[ASAP] Regioselectivity in Diels–Alder Cycloadditions of <sup>#6094</sup>C<sub>68</sub> Fullerene with a Triplet Ground State (Fri, 28 Jun 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b00921
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