The Journal of Organic Chemistry



[ASAP] Indole-Fused Acridone: Synthesis, Structures, Proton Transfer, and Hole-Transport Properties (Thu, 21 Mar 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.8b02939
>> Read More

[ASAP] Asymmetric Synthesis of ?-Hydroxy Pinacolboronates through Copper-Catalyzed Enantioselective Hydroboration of a,ß-Unsaturated Aldehydes (Thu, 21 Mar 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.8b03045
>> Read More

[ASAP] Enantioselective Synthesis of 3,4-Dihydropyrimidin-2(1<italic toggle="yes">H</italic>)-ones through Organocatalytic Transfer Hydrogenation of 2-Hydroxypyrimidines (Thu, 21 Mar 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.8b03128
>> Read More

[ASAP] Aspergiolides A and B: Core Structural Establishment and Synthesis of Structural Analogues (Thu, 21 Mar 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.8b03185
>> Read More

[ASAP] Diastereoselective ABB' Three-Component Synthesis of Highly Functionalized Spirooxindoles Bearing Five Consecutive Asymmetric Carbons (Thu, 21 Mar 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.8b03270
>> Read More

[ASAP] Oligosaccharide Sensing in Aqueous Media Using Porphyrin–Curdlan Conjugates: An Allosteric Signal-Amplification System (Thu, 21 Mar 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b00040
>> Read More

[ASAP] One-Pot Oxidative Coupling/Decyanation of 6,7-Diphenylindolizine-5-carbonitriles and 2,3-Diphenylquinolizine-4-carbonitriles (Thu, 21 Mar 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b00041
>> Read More

[ASAP] Achieving Nickel Catalyzed C–S Cross-Coupling under Mild Conditions Using Metal–Ligand Cooperativity (Thu, 21 Mar 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b00075
>> Read More

[ASAP] Synthesis of 4-Sulfenyl Isoxazoles through AlCl<sub>3</sub>-Mediated Electrophilic Cyclization and Sulfenylation of 2-Alkyn-1-one <italic toggle="yes">O</italic>-Methyloximes (Thu, 21 Mar 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b00256
>> Read More

[ASAP] Pyridine-Fused 2-Pyridones via Povarov and A<sup>3</sup> Reactions: Rapid Generation of Highly Functionalized Tricyclic Heterocycles Capable of Amyloid Fibril Binding (Wed, 20 Mar 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.8b03015
>> Read More

[ASAP] Unusual Formation of Cyclopenta[<italic toggle="yes">b</italic>]indoles from 3-Indolylmethanols and Alkynes (Wed, 20 Mar 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.8b03027
>> Read More

[ASAP] “On Water” Direct Organocatalytic Cyanoarylmethylation of Isatins for the Diastereoselective Synthesis of 3-Hydroxy-3-cyanomethyl Oxindoles (Wed, 20 Mar 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.8b03194
>> Read More

[ASAP] Theoretical Investigation of the Enantioselective [4 + 2] Cycloaddition Reaction of <italic toggle="yes">o</italic>-Hydroxystyrene and Azlactone (Wed, 20 Mar 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b00032
>> Read More

[ASAP] Access to 27-Nortomatidine and 27-Norsoladulcidine Derivatives (Wed, 20 Mar 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b00103
>> Read More

[ASAP] Regiospecific Cleavage of S–N Bonds in Sulfonyl Azides: Sulfonyl Donors (Tue, 19 Mar 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.8b03046
>> Read More

[ASAP] Boron-Catalyzed Azide Insertion of a-Aryl a-Diazoesters (Tue, 19 Mar 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.8b03278
>> Read More

[ASAP] Diselenide Bonds as an Alternative to Outperform the Efficiency of Disulfides in Self-Healing Materials (Tue, 19 Mar 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b00014
>> Read More

[ASAP] Transition-Metal-Free Oxidation of Benzylic C–H Bonds of Six-Membered N-Heteroaromatic Compounds (Tue, 19 Mar 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b00035
>> Read More

[ASAP] Sulfur-Mediated Electrophilic Cyclization of Aryl-Substituted Internal Alkynes (Tue, 19 Mar 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b00136
>> Read More

[ASAP] Iodine(III)-Mediated, Controlled Di- or Monoiodination of Phenols (Tue, 19 Mar 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b00161
>> Read More

[ASAP] Functionalized Helical ß-Peptoids (Tue, 19 Mar 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b00218
>> Read More

[ASAP] 1,3-Dipolar Cycloaddition of Isatin-Derived Azomethine Ylides with 2<italic toggle="yes">H</italic>-Azirines: Stereoselective Synthesis of 1,3-Diazaspiro[bicyclo[3.1.0]hexane]oxindoles (Tue, 19 Mar 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b00242
>> Read More

[ASAP] Halo-1,2,3-triazolium Salts as Halogen Bond Donors for the Activation of Imines in Dihydropyridinone Synthesis (Tue, 19 Mar 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b00248
>> Read More

[ASAP] KOAc-Catalyzed One-Pot Three-Component 1,3-Dipolar Cycloaddition of a-Diazo Compounds, Nitrosoarenes, and Alkenes: An Approach to Functionalized Isoxazolidines (Tue, 19 Mar 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b00299
>> Read More

[ASAP] Amination of Carbenium Ions Generated by Directed Protonolysis of Cyclopropane (Mon, 18 Mar 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.8b02576
>> Read More

[ASAP] Nucleophilic Organic Base DABCO-Mediated Chemospecific Meinwald Rearrangement of Terminal Epoxides into Methyl Ketones (Mon, 18 Mar 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.8b03171
>> Read More

[ASAP] Divergent Synthesis of 1,2-Benzo[<italic toggle="yes">e</italic>]thiazine and Benzo[<italic toggle="yes">d</italic>]thiazole Analogues Containing a <italic toggle="yes">S</italic>-Trifluoromethyl Sulfoximine Group: Preparation and New Properties of the Adachi Reagent (Mon, 18 Mar 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b00079
>> Read More

[ASAP] Ir-Catalyzed C–H Amidation and Borylation of Anthraquinones (Mon, 18 Mar 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b00106
>> Read More

[ASAP] Factors Controlling the Reactivity of Strained-Alkyne Embedded Cycloparaphenylenes (Mon, 18 Mar 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b00292
>> Read More

[ASAP] Visible-Light-Promoted Three-Component Coupling Annulation: Synthesis of 2-Iminothiazolidin-4-ones via in Situ Formed Electron Donor–Acceptor Complexes (Mon, 18 Mar 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b00305
>> Read More

[ASAP] Correction to Metal-Free Regioselective Monocyanation of Hydroxy-, Alkoxy-, and Benzyloxyarenes by Potassium Thiocyanate and Silica Sulfuric Acid as a Cyanating Agent (Mon, 18 Mar 2019)
The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b00656
>> Read More

[ASAP] Transition-Metal-Free One-Step Synthesis of Ynamides (Fri, 15 Mar 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.8b03192
>> Read More

[ASAP] Formal [4 + 2] Annulation of Oxindole-Embedded <italic toggle="yes">ortho</italic>-Quinone Methides with 1,3-Dicarbonyls: Synthesis of Spiro[Chromen-4,3'-Oxindole] Scaffolds (Fri, 15 Mar 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.8b03260
>> Read More

[ASAP] Transfer of Sequence Information and Replication of Diimine Duplexes (Fri, 15 Mar 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b00095
>> Read More

[ASAP] External Oxidant-Dependent Reactivity Switch in Copper-Mediated Intramolecular Carboamination of Alkynes: Access to a Different Class of Fluorescent Ionic Nitrogen-Doped Polycyclic Aromatic Hydrocarbons (Fri, 15 Mar 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b00120
>> Read More

[ASAP] Bonded to Carbon or Nitrogen? This is a Question on the Regioselectivity in Hyperconjugative Aromaticity (Thu, 14 Mar 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.8b02996
>> Read More

[ASAP] Aerobic and Ligand-Free Manganese-Catalyzed Homocoupling of Arenes or Aryl Halides via in Situ Formation of Aryllithiums (Wed, 13 Mar 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.8b02834
>> Read More

[ASAP] Pd-Catalyzed Four-Component Sequential Reaction Delivers a Modular Fluorophore Platform for Cell Imaging (Wed, 13 Mar 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.8b02845
>> Read More

[ASAP] Tiara[<italic toggle="yes">n</italic>]uril: A Glycoluril-Based Macrocyclic Host with Cationic Walls (Wed, 13 Mar 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.8b02913
>> Read More

[ASAP] Regioselective Photocycloaddition of Saccharin Anion to p-Systems: Continuous-Flow Synthesis of Benzosultams (Wed, 13 Mar 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.8b02984
>> Read More

[ASAP] Chemoselective Carbonyl Allylations with Alkoxyallylsiletanes (Wed, 13 Mar 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.8b03028
>> Read More

[ASAP] <italic toggle="yes">exo/endo</italic> Selectivity Control in Diels–Alder Reactions of Geminal Bis(silyl) Dienes: Theoretical and Experimental Studies (Wed, 13 Mar 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.8b03090
>> Read More

[ASAP] <italic toggle="yes">Meso</italic>-Substituent-Directed Aggregation Behavior and Water Solubility: Direct Functionalization of Methine Chain in Thiazole Orange and Biological Applications in Aqueous Buffer (Wed, 13 Mar 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.8b03122
>> Read More

[ASAP] Palladium Catalyzed Regioselective Synthesis of Substituted Biaryl Amides through Decarbonylative Arylation of Phthalimides (Wed, 13 Mar 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.8b03157
>> Read More

[ASAP] Desymmetrization by Asymmetric Copper-Catalyzed Intramolecular C–H Insertion Reactions of a-Diazo-ß-oxosulfones (Wed, 13 Mar 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.8b03160
>> Read More

[ASAP] AgSCF<sub>3</sub>/Na<sub>2</sub>S<sub>2</sub>O<sub>8</sub>-Promoted Trifluoromethylthiolation/Cyclization of <italic toggle="yes">o</italic>-Propargyl Arylazides/<italic toggle="yes">o</italic>-Alkynyl Benzylazides: Synthesis of SCF<sub>3</sub>-Substituted Quinolines and Isoquinolines (Wed, 13 Mar 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b00181
>> Read More

[ASAP] Synthesis of Divergent Benzo[<italic toggle="yes">b</italic>]fluorenones through Cycloaromatization Reactions of 1,5-Enynols and 1,5-Diynols (Wed, 13 Mar 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b00231
>> Read More

[ASAP] C<sub>2</sub>-Symmetric Chiral Squaramide, Recyclable Organocatalyst for Asymmetric Michael Reactions (Wed, 13 Mar 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b00252
>> Read More

[ASAP] Mn(II)-Catalyzed C–H Alkylation of Imidazopyridines and <italic toggle="yes">N</italic>-Heteroarenes via Decarbonylative and Cross-Dehydrogenative Coupling (Wed, 13 Mar 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b00366
>> Read More

[ASAP] Investigation of a Weak Temperature–Rate Relationship in the Carbamoylation of a Barbituric Acid Pharmaceutical Intermediate (Wed, 13 Mar 2019)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b00411
>> Read More