The Journal of Organic Chemistry



[ASAP] Synthesis of Dibenzosuberones Bearing an Isoxazole Group via Palladium-Catalyzed Intramolecular C–H/C–Br Bond Cross-Coupling of Ortho-Aroylated 3,5-Diarylisoxazoles (Fri, 03 Apr 2020)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.0c00346
>> Read More

[ASAP] DABCO-Catalyzed Michael/Alkylation Cascade Reactions Involving a-Substituted Ammonium Ylides for the Construction of Spirocyclopropyl Oxindoles: Access to the Powerful Chemical Leads against HIV-1 (Fri, 03 Apr 2020)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b03164
>> Read More

[ASAP] Catalytic Asymmetric Diarylphosphine Addition to a-Diazoesters for the Synthesis of P-Stereogenic Phosphinates via P*—N Bond Formation (Fri, 03 Apr 2020)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.0c00181
>> Read More

[ASAP] Toward FAIRness and a User-Friendly Repository for Supporting NMR Data (Fri, 03 Apr 2020)
The Journal of Organic Chemistry DOI: 10.1021/acs.joc.0c00800
>> Read More

[ASAP] Direct Photorelease of Alcohols from Boron-Alkylated BODIPY Photocages (Fri, 03 Apr 2020)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.0c00044
>> Read More

[ASAP] Photoredox-Catalyzed Oxy-/Aminofluoroalkylative Cyclization of Alkenes (Fri, 03 Apr 2020)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.0c00457
>> Read More

[ASAP] Catalytic Asymmetric [4 + 2] Cycloaddition of <italic toggle="yes">ortho</italic>-Alkenyl Naphthols/Phenols with <italic toggle="yes">ortho</italic>-Quinone Methides: Highly Stereoselective Synthesis of Chiral 2,3,4-Trisubstituted Chromans (Fri, 03 Apr 2020)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b03302
>> Read More

[ASAP] Does the Reaction of Cyclopropyl Acid Chlorides and Imines To Form 1,3-Oxazin-4-enone Heterocycles Proceed via a Ketene or an <italic toggle="yes">N</italic>-Acyl-iminium Mechanism? (Thu, 02 Apr 2020)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.0c00229
>> Read More

[ASAP] Synthesis of Cross-Conjugated Polyenes via Palladium-Catalyzed Oxidative C–C Bond Forming Cascade Reactions of Allenes (Thu, 02 Apr 2020)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.0c00186
>> Read More

[ASAP] Access to (<italic toggle="yes">Z</italic>)-1,2-Endiamides and 1,1-Endiamides via a Base-Promoted Tandem Reaction (Thu, 02 Apr 2020)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b03305
>> Read More

[ASAP] Acyl Cyanides as Bifunctional Reagent: Application in Copper-Catalyzed Cyanoamidation and Cyanoesterification Reaction (Thu, 02 Apr 2020)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b03500
>> Read More

[ASAP] Access to Fused Pyrroles from Cyclic 1,3-Dienyl Boronic Esters and Arylnitroso Compounds (Thu, 02 Apr 2020)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b03214
>> Read More

[ASAP] Correction to “One-Pot Generation of Functionalized Benzynes from Readily Available 2-Hydroxyphenylboronic Acids” (Wed, 01 Apr 2020)
The Journal of Organic Chemistry DOI: 10.1021/acs.joc.0c00719
>> Read More

[ASAP] Reaction Cycling for Kinetic Analysis in Flow (Wed, 01 Apr 2020)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.0c00216
>> Read More

[ASAP] A Catalytic Dual Isomerization/Allylboration Sequence for the Stereoselective Construction of Congested Secondary Homoallylic Alcohols (Wed, 01 Apr 2020)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.0c00565
>> Read More

[ASAP] Metal-Free Oxidative Esterification of Ketones and Potassium Xanthates: Selective Synthesis of a-Ketoesters and Esters (Wed, 01 Apr 2020)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b03272
>> Read More

[ASAP] Synthesis of Triarylmethanes by Decarbonylation of 3,3-Diaryl Benzofuranones (Wed, 01 Apr 2020)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b03433
>> Read More

[ASAP] Fungal Light Emitter: Understanding Its Chemical Nature and pH-Dependent Emission in Water Solution (Wed, 01 Apr 2020)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.0c00246
>> Read More

[ASAP] Photoelectrocyclization Reactions of Conjugated Cycloalkenones: Scope and Reactivity (Wed, 01 Apr 2020)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.0c00197
>> Read More

[ASAP] C–H Sulfonylation via 1,3-Rearrangement of Sulfonyl Group in <italic toggle="yes">N</italic>-Protected 3-Bis-sulfonimidoindole Derivatives Using Fluorine Reagent (Wed, 01 Apr 2020)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b03498
>> Read More

[ASAP] Gentianelloids A and B: Immunosuppressive 10,11-<italic toggle="yes">seco</italic>-Gentianellane Sesterterpenoids from the Traditional Uighur Medicine <italic toggle="yes">Gentianella turkestanorum</italic> (Wed, 01 Apr 2020)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.0c00272
>> Read More

[ASAP] Enantioselective Synthesis of 3,4-Dihydropyran-2-ones via Phase-Transfer-Catalyzed Addition–Cyclization of Acetylacetone to Cinnamic Thioesters (Wed, 01 Apr 2020)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b03216
>> Read More

[ASAP] Diels–Alder/Ene Reactivities of 2-(1'-Cycloalkenyl)thiophenes and 2-(1'-Cycloalkenyl)benzo[<italic toggle="yes">b</italic>]thiophenes with <italic toggle="yes">N</italic>-Phenylmaleimides: Role of Cycloalkene Ring Size on Benzothiophene and Dibenzothiophene Product Distributions (Tue, 31 Mar 2020)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b03363
>> Read More

[ASAP] Bringing a Molecular Plus One: Synergistic Binding Creates Guest-Mediated Three-Component Complexes (Tue, 31 Mar 2020)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.0c00220
>> Read More

[ASAP] Synthesis of Sulfones <italic toggle="yes">via</italic> Ru(II)-Catalyzed Sulfination of Boronic Acids (Tue, 31 Mar 2020)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b03403
>> Read More

[ASAP] Synthesis of Functionalized Isoindolinones via Calcium Catalyzed Generation and Trapping of <italic toggle="yes">N</italic>-Acyliminium Ions (Tue, 31 Mar 2020)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.0c00482
>> Read More

[ASAP] Allylboration of Ketones and Imines with a Highly Reactive Bifunctional Allyl Pinacolatoboronate Reagent (Tue, 31 Mar 2020)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b03222
>> Read More

[ASAP] Visible-Light-Mediated [2+2+1] Carbocyclization Reactions of 1,7-Enynes with Bromofluoroacetate to Form Fused Monofluorinated Cyclopenta[<italic toggle="yes">c</italic>]quinolin-4-ones (Tue, 31 Mar 2020)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.0c00087
>> Read More

[ASAP] 5-Aryltetrazoles from Direct C–H Arylation with Aryl Bromides (Tue, 31 Mar 2020)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.0c00085
>> Read More

[ASAP] Weak Coordinating Carbonyl-Directed Rhodium(III)-Catalyzed C–H Activation at the C4-Position of Indole with Allyl Alcohols (Tue, 31 Mar 2020)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.0c00277
>> Read More

[ASAP] Thiourea Derivative of 2-[(1<italic toggle="yes">R</italic>)-1-Aminoethyl]phenol: A Flexible Pocket-like Chiral Solvating Agent (CSA) for the Enantiodifferentiation of Amino Acid Derivatives by NMR Spectroscopy (Mon, 30 Mar 2020)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.0c00027
>> Read More

[ASAP] Catalyst-Free Conjugate Addition of Indolizines to <italic toggle="yes">In Situ</italic>-Generated Oxidized Morita–Baylis–Hillman Adducts (Mon, 30 Mar 2020)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.0c00189
>> Read More

[ASAP] Structure–Property Relationships in Unsymmetric Bis(antiaromatics): Who Wins the Battle between Pentalene and Benzocyclobutadiene?<xref rid="notes-2" ref-type="statement">†</xref> (Mon, 30 Mar 2020)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b03119
>> Read More

[ASAP] Synthesis of 8-Alkoxy-5<italic toggle="yes">H</italic>-isochromeno[3,4-<italic toggle="yes">c</italic>]isoquinolines and 1-Alkoxy-4-arylisoquinolin-3-ols through Rh(III)-Catalyzed C–H Functionalization of Benzimidates with 4-Diazoisochroman-3-imines and 4-Diazoisoquinolin-3-ones (Mon, 30 Mar 2020)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.0c00283
>> Read More

[ASAP] Total Synthesis of Nominal <italic toggle="yes">ent</italic>-Chlorabietol B (Mon, 30 Mar 2020)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.0c00233
>> Read More

[ASAP] Cobalt-Catalyzed One-Step Access to Pyroquilon and C-7 Alkenylation of Indoline with Activated Alkenes Using Weakly Coordinating Functional Groups (Fri, 27 Mar 2020)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.0c00023
>> Read More

[ASAP] Access to Phenothiazine Derivatives via Iodide-Mediated Oxidative Three-Component Annulation Reaction (Fri, 27 Mar 2020)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.0c00562
>> Read More

[ASAP] One-Pot Amberlyst 15-Controlled Cyclocondensation of Piperidines and Arylaldehydes: Synthesis of 3,5-Diarylmethylpyridines (Fri, 27 Mar 2020)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b03315
>> Read More

[ASAP] Late-Stage Conversion of a Metabolically Labile Aryl Methyl Ether-Containing Natural Product to Fluoroalkyl Analogues (Fri, 27 Mar 2020)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.0c00125
>> Read More

[ASAP] Pd/C-Catalyzed Carbonylative Synthesis of a-Carbonyl-a'-Amide Sulfoxonium Ylides from Azides (Fri, 27 Mar 2020)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.0c00273
>> Read More

[ASAP] Asymmetric Synthesis of a Key Dextromethorphan Intermediate and Its Analogues Enabled by a New Cyclohexylamine Oxidase: Enzyme Discovery, Reaction Development, and Mechanistic Insight (Fri, 27 Mar 2020)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.0c00469
>> Read More

[ASAP] Visible- and UV-Light-Induced Decarboxylative Radical Reactions of Benzoic Acids Using Organic Photoredox Catalysts (Tue, 24 Mar 2020)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.0c00055
>> Read More

[ASAP] Twisting and Turning the Sulfonamide Bond: A Synthetic, Quantum Chemical, and Crystallographic Study (Tue, 24 Mar 2020)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b03394
>> Read More

[ASAP] Synthesis of Diaryl Hydroxyl Dicarboxylic Acids from Amino Acids (Tue, 10 Mar 2020)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b03320
>> Read More

[ASAP] Carbonyl-Stabilized Phosphorus Ylide as an Organocatalyst for Cyanosilylation Reactions Using TMSCN (Mon, 09 Mar 2020)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b03347
>> Read More

[ASAP] Reworking Organic Synthesis for the Modern Age: Synthetic Strategies Based on Continuous-Flow Addition and Condensation Reactions with Heterogeneous Catalysts (Mon, 02 Mar 2020)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b03416
>> Read More

[ASAP] Aspects of Phosphaallene Chemistry: Heat-Induced Formation of 1,2-Dihydrophosphetes by Intramolecular Nucleophilic Aromatic Substitution and Photochemical Generation of Tricyclic Phosphiranes (Thu, 27 Feb 2020)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b03056
>> Read More

[ASAP] Synthesis of Highly Fused Pyrano[2,3-<italic toggle="yes">b</italic>]pyridines via Rh(III)-Catalyzed C–H Activation and Intramolecular Cascade Annulation under Room Temperature (Tue, 25 Feb 2020)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b03102
>> Read More

[ASAP] Reactivity of Boronic Acids toward Catechols in Aqueous Solution (Fri, 31 Jan 2020)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b03326
>> Read More

[ASAP] Axial Chirality around N–P Bonds Induced by Complexation between E(C<sub>6</sub>F<sub>5</sub>)<sub>3</sub> (E = B, Al) and an <italic toggle="yes">N</italic>-Phosphine Oxide-Substituted Imidazolinylidene: A Key Intermediate in the Catalytic Phosphinoylation of CO<sub>2</sub> (Fri, 10 Jan 2020)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.9b03210
>> Read More