The Journal of Organic Chemistry

High-Yielding Syntheses of Crown Ether-Based Pyridyl Cryptands (Wed, 26 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01389
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Synthesis and Characterization of Contorted Pentabenzo-Fused Coronenes as Semiconducting Materials (Wed, 26 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01328
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Preparation of 3-Iodoquinolines from N-Tosyl-2-propynylamines with Diaryliodonium Triflate and N-Iodosuccinimide (Wed, 26 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01433
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Synthesis of a 3-Amino-2,3-dihydropyrid-4-one and Related Heterocyclic Analogues as Mechanism-Based Inhibitors of BioA, a Pyridoxal Phosphate-Dependent Enzyme (Wed, 26 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b00847
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Diastereoselective Construction of the 6-Oxa-2-azabicyclo[3.2.1]octane Scaffold from Chiral α-Hydroxyaldehyde Derivatives by the Aza-Prins Reaction (Wed, 26 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01291
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Organocatalytic Asymmetric Mannich/Aza-Michael Cascade Reaction of δ-Formyl-α,β-unsaturated Ketones with Cyclic N-Sulfimines: Enantioselective Synthesis of Benzosulfamidate-Fused Pyrrolidines (Tue, 25 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01533
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Synthesis of 2-Amino-3-hydroxy-3H-indoles via Palladium-Catalyzed One-Pot Reaction of Isonitriles, Oxygen, and N-Tosylhydrazones Derived from 2-Acylanilines (Tue, 25 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01195
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Synthesis and Evaluation of Agelastatin Derivatives as Potent Modulators for Cancer Invasion and Metastasis (Tue, 25 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01162
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Metal-Free Three-Component Regioselective Aminofluorination of Styrene Derivatives (Tue, 25 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01089
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Investigation and Demonstration of Catalyst/Initiator-Driven Selectivity in Thiol-Michael Reactions (Tue, 25 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01200
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Indolylmethanols as Reactants in Catalytic Asymmetric Reactions (Mon, 24 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01458
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The Synthesis of Certain Derivatives and Analogues of (−)- and (+)-Galanthamine and an Assessment of their Capacities to Inhibit Acetylcholine Esterase (Mon, 24 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01062
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Synthesis of (±)-Aphanorphine Using Rh-Catalyzed Cyclohydrocarbonylation (Mon, 24 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b00923
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Hypervalent Iodine-Mediated Oxidative Rearrangement of N–H Ketimines: An Umpolung Approach to Amides (Mon, 24 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01468
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Preparation of Quinazolines via a 2+2+2 Annulation from Aryldiazonium Salts and Nitriles (Mon, 24 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01325
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Cycloaddition Reactions of Cobalt-Complexed Macrocyclic Alkynes: The Transannular Pauson–Khand Reaction (Mon, 24 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01369
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Pd(II)/Bipyridine-Catalyzed Conjugate Addition of Arylboronic Acids to α,β-Unsaturated Carboxylic Acids. Synthesis of β-Quaternary Carbons Substituted Carboxylic Acids (Mon, 24 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01248
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Synthesis of Oxatricyclooctanes via Photoinduced Intramolecular Oxa-[4+2] Cycloaddition of Substituted o-Divinylbenzenes (Mon, 24 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01055
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Ethynylene-linked Figure-Eight Octaphyrin(1.2.1.1.1.2.1.1): Synthesis and Characterization of Its Two Oxidation States (Fri, 21 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01592
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Lithium Amide Protected against Hydrolysis by Aggregated Lithium Halides: An MS + DFT Investigation (Fri, 21 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01419
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Origins of Stereoselectivity of Enamine–Iminium-Activated Nazarov Cyclizations by Vicinal Diamines (Fri, 21 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01606
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Synthesis and Structures of Zigzag Shaped [12]Cyclo-p-phenylene Composed of Dinaphthofuran Units and Biphenyl Units (Thu, 20 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01053
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Pd-Catalyzed/Iodide-Promoted α-Arylation of Ketones for the Regioselective Synthesis of Isocoumarins (Thu, 20 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01355
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Studies on the Photochemical Rearrangements of Enantiomerically Pure, Polysubstituted, and Variously Annulated Bicyclo[2.2.2]octenones (Thu, 20 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01243
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Pd-Catalyzed Carbonylative Carboperfluoroalkylation of Alkynes. Through-Space 13C–19F Coupling as a Probe for Configuration Assignment of Fluoroalkyl-Substituted Olefins (Thu, 20 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01236
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NHC-Cu(I)-Catalyzed Friedländer-Type Annulation of Fluorinated o-Aminophenones with Alkynes on Water: Competitive Base-Catalyzed Dibenzo[b,f][1,5]diazocine Formation (Thu, 20 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01235
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Fluorescence Enhancement of Unconstrained GFP Chromophore Analogues Based on the Push–Pull Substituent Effect (Thu, 20 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01260
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Interplay of Conformational and Chemical Transformations of Ortho-Substituted Aromatic Nitroso Oxides: Experimental and Theoretical Study (Thu, 20 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b00537
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Palladium-Catalyzed Intermolecular Oxidative Cyclization of Allyltosylamides with AcOH: Assembly of 3-Pyrrolin-2-ones (Thu, 20 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b00804
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Flow Synthesis of Diaryliodonium Triflates (Thu, 20 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01346
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Structure–Reactivity Relationships of Conformationally Armed Disaccharide Donors and Their Use in the Synthesis of a Hexasaccharide Related to the Capsular Polysaccharide from Streptococcus pneumoniae Type 37 (Wed, 19 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01264
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Total Synthesis of Lycopladine A and Carinatine A via a Base-Mediated Carbocyclization (Wed, 19 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b00908
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Synthesis and Structural Revision of the Fungal Tetramic Acid Metabolite Spiroscytalin (Wed, 19 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b00727
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Cu-Catalyzed Aminodifluoroalkylation of Alkynes and α-Bromodifluoroacetamides (Wed, 19 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01313
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Factors Governing the Diels–Alder Reactivity of (2,7)Pyrenophanes (Wed, 19 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01449
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Solvolytic Behavior of Aryl and Alkyl Carbonates. Impact of the Intrinsic Barrier on Relative Reactivities of Leaving Groups (Wed, 19 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b00885
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Total Synthesis of Cardiolipins Containing Chiral Cyclopropane Fatty Acids (Wed, 19 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b00945
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Cobalt(II)-Catalyzed Isocyanide Insertion Reaction with Sulfonyl Azides in Alcohols: Synthesis of Sulfonyl Isoureas (Wed, 19 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01127
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Synthesis of Spiro[indazole-3,3′-indolin]-2′-ones via [3 + 2] Dipolar Cycloaddition of Arynes with 3-Diazoindolin-2-ones and Indazolo[2,3-c]quinazolin-6(5H)-ones by Subsequent Thermal Isomerization (Wed, 19 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b00990
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Diastereoselective Synthesis of CF3-Containing Vicinal Diamines (Wed, 19 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01261
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Pathways in the Degradation of Geminal Diazides (Wed, 19 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01019
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Matsutakone and Matsutoic Acid, Two (Nor)steroids with Unusual Skeletons from the Edible Mushroom Tricholoma matsutake (Wed, 19 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01230
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Pyridine–Spiropyran Derivative as a Persistent, Reversible Photoacid in Water (Wed, 19 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01268
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Direct Catalytic Asymmetric Aldol Addition of an α-CF3 Amide to Arylglyoxal Hydrates (Wed, 19 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01381
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Hypervalent Iodine(III)-Promoted Phenyl Transfer Reaction from Phenyl Hydrazides to Nitriles (Wed, 19 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01215
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Approach to the Synthesis of 2,3-Disubstituted-3H-quinazolin-4-ones Mediated by Ph3P–I2 (Wed, 19 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01322
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Synthesis of Thieno-Fused Five- and Six-Membered Nitrogen and Oxygen Heterocycles via Intramolecular Heteroannulation of 4,5-Substituted 3-Amino or 3-Hydroxy 2-Functionalized Thiophenes (Tue, 18 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01153
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Nucleophile-Mediated Ring Expansion of 5-Acyl-substituted 4-Mesyloxymethyl-1,2,3,4-tetrahydropyrimidin-2-ones in the Synthesis of 7-Membered Analogues of Biginelli Compounds and Related Heterocycles (Tue, 18 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01348
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Correction to “Chemical Dynamic Thermodynamic Resolution and S/R Interconversion of Unprotected Unnatural Tailor-made α-Amino Acids” (Tue, 18 Jul 2017)
The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01660
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Highly Fluorescent Red-Light Emitting Bis(boranils) Based on Naphthalene Backbone (Tue, 18 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01001
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Corey–Chaykovsky Reactions of Nitro Styrenes Enable cis-Configured Trifluoromethyl Cyclopropanes (Mon, 17 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b00951
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Perfluorinated and Half-Fluorinated Rubrenes: Synthesis and Crystal Packing Arrangements (Mon, 17 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01383
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Regioselective Diversification of 2,1-Borazaronaphthalenes: Unlocking Isosteric Space via C–H Activation (Mon, 17 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01331
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Total Synthesis of (−)-Chanoclavine I and an Oxygen-Substituted Ergoline Derivative (Mon, 17 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b00573
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Nitroalkenes as Latent 1,2-Biselectrophiles – A Multicatalytic Approach for the Synthesis of 1,4-Diketones and Their Application in a Four-Step One-Pot Reaction to Polysubstituted Pyrroles (Mon, 17 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b00830
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C1′-Azacycloalkyl Hexahydrocannabinols (Mon, 17 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b00988
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Photocatalytic E → Z Isomerization of Polarized Alkenes Inspired by the Visual Cycle: Mechanistic Dichotomy and Origin of Selectivity (Mon, 17 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01281
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Combined Experimental and Computational Study on Ruthenium(II)-Catalyzed Reactions of Diynes with Aldehydes and N,N-Dimethylformamide (Fri, 14 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01229
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Regioselective Synthesis of 2-Vinylanilines Using O-aroyloxycarba-mates by Sequential Decarboxylation/Amination/Heck Reaction (Fri, 14 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01020
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Reversible Multistimuli Switching of a Spiropyran-Functionalized Organic Cage in Solid and Solution (Fri, 14 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b00722
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Mixed Phenyl and Thiophene Oligomers for Bridging Nitronyl Nitroxides (Fri, 14 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b00435
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Synthesis of 1-Azaanthraquinone: Sequential C–N Bond Formation/Lewis Acid Catalyzed Intramolecular Cyclization Strategy (Fri, 14 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01427
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A Tetramer Derived from Islet Amyloid Polypeptide (Fri, 14 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01116
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Mechanistic Studies of Formal Thioboration Reactions of Alkynes (Fri, 14 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01500
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Palladium-Mediated Synthesis of a Near-Infrared Fluorescent K+ Sensor (Fri, 14 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b00845
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Synthesis, Thermodynamic Properties, and Crystal Structure of RNA Oligonucleotides Containing 5-Hydroxymethylcytosine (Fri, 14 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01171
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Decoding the Mechanism of Intramolecular Cu-Directed Hydroxylation of sp3 C–H Bonds (Fri, 14 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01069
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Laterally π-Extended Dithia[6]helicenes with Heptagons: Saddle-Helix Hybrid Molecules (Wed, 12 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01540
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Hypervalent Iodine/HF Reagents for the Synthesis of 3-Fluoropyrrolidines (Tue, 11 Jul 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01266
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Hypervalent Iodine(III)-Mediated Decarboxylative Ritter-Type Amination Leading to the Production of α-Tertiary Amine Derivatives (Tue, 27 Jun 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01202
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Powerful, Thermally Stable, One-Pot-Preparable, and Recyclable Electrophilic Trifluoromethylating Agents: 2,8-Difluoro- and 2,3,7,8-Tetrafluoro-S-(trifluoromethyl)dibenzothiophenium Salts (Thu, 22 Jun 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b00669
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Peptidyl-Prolyl Model Study: How Does the Electronic Effect Influence the Amide Bond Conformation? (Wed, 21 Jun 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b00803
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Regioselective Rh-Catalyzed Hydroformylation of 1,1,3-Trisubstituted Allenes Using BisDiazaPhos Ligand (Mon, 19 Jun 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01140
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Hypervalent-Iodine-Mediated Formation of Epoxides from Carbon(sp2)–Carbon(sp3) Single Bonds (Thu, 15 Jun 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b00883
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Initiation in Photoredox C–H Functionalization Reactions. Is Dimsyl Anion a Key Ingredient? (Tue, 06 Jun 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b00822
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Enantioselective C–C Bond Formation during the Oxidation of 5-Phenylpent-2-enyl Carboxylates with Hypervalent Iodine(III) (Mon, 05 Jun 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b01141
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Perfluoroalkylation of Aryl-N,N-dimethyl Hydrazones Using Hypervalent Iodine(III) Reagents or Perfluoroalkyl Iodides (Thu, 01 Jun 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b00934
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Rhodium(III)-Catalyzed C–H Alkynylation of Ferrocenes with Hypervalent Iodine Reagents (Tue, 09 May 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.7b00775
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Synthesis of Small-Molecule/DNA Hybrids through On-Bead Amide-Coupling Approach (Mon, 20 Mar 2017)
TOC Graphic The Journal of Organic Chemistry DOI: 10.1021/acs.joc.6b02942
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