WO2010003624 heterocyclic compounds, processes for their preparation, medicaments comprising these compounds, and the use thereof

WO2010003624.pdf
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Biological target:

Acetyl-CoA carboxylase: ACC

Activity:

Inhibitor

Steps Conditions Reactions
a Cs2CO3 / DMF Ether synthesis (Nucleophilic substitution)
b Cs2CO3 / DMF Ether synthesis (Nucleophilic substitution)
Steps Conditions Reactions
a Cs2CO3 / KI / DMF Ether synthesis (Nucleophilic substitution)
b DiBAL / toluene Hydrolyl synthesis (Ester reduction)
c APTS / toluene Ether synthesis

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