PATENTSCOPE: EN_ALL:nmr AND PA:teva

RIBOCICLIB SALTS AND SOLID STATE FORMS THEREOF (Fri, 01 Mar 2019)
The present disclosure relates to Ribociclib solid state forms, Ribociclib salts including Ribociclib succinate and solid state forms thereof, as well as processes for preparation thereof and pharmaceutical compositions thereof.
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PROCESSES FOR THE PREPARATION OF NIRAPARIB AND INTERMEDIATES THEREOF (Fri, 22 Feb 2019)
The present invention relates to novel procedures and novel intermediates useful in the synthesis of Niraparib or any salt thereof.
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SALTS AND SOLID STATE FORMS OF PLINABULIN (Fri, 08 Feb 2019)
The present disclosure relates to Plinabulin solid state forms, Plinabulin salts including hydrochloride and solid state forms thereof, processes for preparation thereof and pharmaceutical compositions thereof.
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IMPROVED PROCESSES FOR THE PREPARATION OF GUADECITABINE AND INTERMEDIATES THEREOF (Fri, 18 Jan 2019)
Described are procedures and intermediates for the preparation of guadecitabine, and guadecitabine salts and solid state forms thereof.
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NEW CRYSTALLINE POLYMORPHS OF BARDOXOLONE METHYL (Fri, 18 Jan 2019)
Disclosed are crystalline polymorphs of Bardoxolone methyl, and pharmaceutical compositions thereof.
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SOLID STATE FORMS OF MIDOSTAURIN (Fri, 14 Sep 2018)
The present disclosure relates to solid state forms of Midostaurin, processes for preparation thereof, pharmaceutical compositions thereof, and use thereof in the treatment of Acute Myelogenous Leukemia (AML) and Aggressive Systemic Mastocytosis. Chemical formula: C35H30N4O4 Molecular mass: 570.64 g/mol
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SOLID STATE FORMS OF RUCAPARIB AND OF RUCAPARIB SALTS (Fri, 03 Aug 2018)
Disclosed are solid state forms of Rucaparib and of Rucaparib salts, and pharmaceutical compositions thereof.
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SOLID STATE FORMS OF SOTAGLIFLOZIN (Fri, 13 Apr 2018)
Disclosed are solid state forms of Sotagliflozin, processes for preparation thereof, and pharmaceutical compositions thereof.
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SOLID STATE FORMS OF VALBENAZINE (Fri, 13 Apr 2018)
Solid state forms of Valbenazine, Valbenazine salts, processes for preparation thereof and pharmaceutical compositions thereof are disclosed. Processes for the preparation of Valbenazine and intermediates in the preparation thereof are further described.
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SOLID STATE FORMS OF LUMATEPERONE DITOSYLATE SALT (Fri, 16 Feb 2018)
Disclosed are solid state forms of lumateperone ditosylate, uses thereof, and pharmaceutical compositions thereof.
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CRYSTALLINE FORM VI OF SELEXIPAG (Fri, 02 Feb 2018)
The present disclosure relates to solid state forms of Selexipag, processes for preparation thereof and pharmaceutical compositions thereof.
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SOLID STATE FORMS OF CRISABOROLE (Fri, 19 Jan 2018)
Solid state forms of Crisaborole and salts thereof, processes for preparation thereof and pharmaceutical compositions thereof are disclosed.
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SOLID STATE FORMS OF PALBOCICLIB DIMESYLATE (Fri, 12 Jan 2018)
Solid state forms of Palbociclib dimesylate, processes for preparation thereof and use thereof for preparation of Palbociclib are disclosed.
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SOLID STATE FORMS OF NERATINIB AND SALTS THEREOF (Fri, 05 Jan 2018)
Solid state forms of Neratinib and salts thereof, processes for preparation thereof and pharmaceutical compositions thereof are disclosed.
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SOLID STATE FORMS OF IXAZOMIB CITRATE (Fri, 29 Dec 2017)
The present disclosure encompasses solid state forms of Ixazomib Citrate and pharmaceutical compositions thereof. Also disclosed are processes for preparation of Ixazomib Citrate.
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ASYMMETRIC SYNTHESIS OF FUNAPIDE (Fri, 22 Dec 2017)
This invention is directed to asymmetric synthesis of funapide, which is useful for the treatment and/or prevention of sodium channel-mediated diseases or conditions, such as pain.
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SOLID STATE FORMS OF NILOTINIB SALTS (Fri, 22 Sep 2017)
The present disclosure relates to solid state forms of Nilotinib fumarate and Nilotinib hydrochloride L-tartaric acid co-crystals, processes for preparation thereof, pharmaceutical compositions thereof, and methods of use thereof.
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SOLID STATE FORMS OF VENETOCLAX AND PROCESSES FOR PREPARATION OF VENETOCLAX (Fri, 15 Sep 2017)
Solid state forms of Venetoclax, pharmaceutical compositions thereof, and uses thereof are disclosed. Also disclosed are processes for the preparation of Venetoclax.
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DIHYDROQUINOLINES AND USES THEREOF (Fri, 14 Jul 2017)
The present invention provides a compound or a pharmaceutically acceptable salt or ester thereof. The present invention also provides a pharmaceutical composition comprising the compound of the present invention and a pharmaceutically acceptable carrier. The present invention also provides a method of treating a subject afflicted with multiple sclerosis comprising administering to the subject an amount of the compound of the present invention.
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SOLID STATE FORMS OF BREXPIPRAZOLE (Fri, 23 Jun 2017)
The present disclosure relates to solid state forms of Brexpiprazole, as well as uses and compositions comprising the solid state forms.
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