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PERINDOPRIL TOSYLATE (Wed, 28 Sep 2011)
The present invention relates to a novel salt of perindopril, namely the paratoluene sulfonic acid salt. The present invention also relates to an amorphous form of the perindopril paratoluene sulfonic acid salt. The invention further relates to processes for the preparation of the novel salt and the amorphous form thereof. The invention also relates to pharmaceutical compositions comprising the perindopril tosylate for the treatment of hypertension and heart failure.
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CRYSTALLINE FORMS OF FEBUXOSTAT (Wed, 28 Dec 2011)
New forms of Febuxostat have been prepared and characterized. These forms are useful, for example, in the chronic management of hyperuricemia in patients with gout.
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Crystalline forms of febuxostat (Wed, 12 Dec 2012)
New forms of Febuxostat have been prepared and characterized. These forms are useful, for example, in the chronic management of hyperuricemia in patients with gout.
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Crystalline form of tigecycline and processes for preparation thereof (Wed, 17 Nov 2010)
The present invention provides a crystalline form of Tigecycline, and methods of for preparation of said crystalline form.
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Crystalline form of tigecycline and processes for preparation thereof (Wed, 06 Oct 2010)
The present invention provides a crystalline form of Tigecycline, and methods of for preparation of said crystalline form.
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Crystal form of 9-hydroxy-risperidone (paliperidone) (Wed, 16 Dec 2009)
The present invention provides a crystalline form of Paliperidone, and processes for preparing thereof.
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SOLID STATE FORMS OF SITAGLIPTIN SALTS (Thu, 14 Oct 2010)
Solid state forms of Sitagliptin salts, processes for preparing the solid state forms, and pharmaceutical composi-tions thereof, are provided.
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Crystalline forms of Febuxostat (Thu, 11 Jul 2013)
New forms of Febuxostat have been prepared and characterized. These forms are useful, for example, in the chronic management of hyperuricemia in patients with gout.
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Crystalline forms of febuxostat (Thu, 19 Sep 2013)
New forms of Febuxostat have bean, prepared and characterized. These forms are useful for examples in the chronic management of hyperuricemia in patients with gout.
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Crystal form of 9-hydroxy-risperidone (paliperidone) (Wed, 16 Dec 2009)
The present invention provides a crystalline form of Paliperidone, and processes for preparing thereof.
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RALTEGRAVIR SALTS AND CRYSTALLINE FORMS THEREOF (Wed, 16 Jan 2013)
The present invention includes new salts of Raltegravir and crystalline forms thereof, pharmaceutical compositions containing the salts or crystalline forms, methods of using the salts or crystalline forms or the compositions to treat HIV infection or to prepare medicament for treating HIV infection, and a process for preparing Raltegravir potassium.
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Solid state forms of sitagliptin salts (Thu, 06 Oct 2011)
Crystalline forms of Sitagliptin salts, processes for preparing crystalline forms of Sitagliptin salts, and pharmaceutical compositions of Sitagliptin salts are provided.
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Raltegravir salts and crystalline forms thereof (Thu, 18 Apr 2013)
The present invention includes new salts of Raltegravir and crystalline forms thereof, pharmaceutical compositions containing the salts or crystalline forms, methods of using the salts or crystalline forms or the compositions to treat HIV infection or to prepare medicament for treating HIV infection, and a process for preparing Raltegravir potassium.
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NILOTINIB HCI CRYSTALLINE FORMS (Wed, 22 Dec 2010)
Crystalline forms of Nilotinib HCl are described. (I)
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CRYSTALLINE FORMS OF FEBUXOSTAT (Thu, 16 Dec 2010)
New forms of Febuxostat have been prepared and characterized. These forms are useful, for example, in the chronic management of hyperuricemia in patients with gout.
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SOLID STATE FORMS OF CABAZITAXEL AND PROCESSES FOR PREPARATION THEREOF (Wed, 29 Jan 2014)
The invention relates to solid state forms of Cabazitaxel, and processes for preparation, via novel synthetic intermediates, thereof, and formulations comprising one or more of the solid state forms of Cabazitaxel. The present invention further provides pharmaceutical compositions comprising one or more of the solid state forms of Cabazitaxel, and a method of treating hormone-refractory prostate cancer.
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Crystalline raltegravir sodium salts (Wed, 29 Oct 2014)
The present invention includes new salts of Raltegravir and crystalline forms thereof, pharmaceutical compositions containing the salts or crystalline forms, methods of using the salts or crystalline forms or the compositions to treat HIV infection or to prepare medicament for treating HIV infection, and a process for preparing Raltegravir potassium.
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Solid state forms of sitagliptin salts (Thu, 30 Sep 2010)
Solid state forms of Sitagliptin salts (e.g. Sitagliptin sulfate, Formula I), processes for preparing the solid state forms, and pharmaceutical compositions thereof, are provided. These compounds are of a class of dipeptidyl peptidase IV enzyme inhibitors which are useful, for example, for the manufacture of a medicament for the treatment of type 2 diabetes mellitus. embedded image
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Process for preparing a polymorphic form of atorvastatin calcium (Wed, 01 Jun 2005)
The present invention relates to atorvastatin calcium, a useful agent for lowering serum cholesterol levels. New atorvastatin calcium Form V, processes for preparing the new form, and pharmaceutical compositions and dosage forms containing the new form are disclosed.
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Crystalline forms of febuxostat (Wed, 28 Nov 2012)
New forms of Febuxostat have been prepared and characterized. These forms are useful, for example, in the chronic management of hyperuricemia in patients with gout.
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